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Roscovitine, Free Base **

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产品名称: Roscovitine, Free Base **
产品型号: LC R-1234
产品展商: 原装进口
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Roscovitine, Free Base **


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Roscovitine, Free Base **

产品名称:Roscovitine, Free Base
产品货号:LC  R-1234
产品规格:10 MG
Roscovitine is a potent inhibitor of p34cdc2 (IC50 = 0.2 µM).  Also inhibits p33cdk2 and p33cdk5.  Havlicek, L., et al.  "Cytokinin-derived cyclin-dependent kinase inhibitors: synthesis and cdc2 inhibitory activity of olomoucine and related compounds."  J. Med. Chem. 40:  408-412 (1997).
NOTE:  The word "Roscovitine" inherently means the R-isomer.
Storage:  Store at or below -20 ºC.  Solubility:  Prepare initial stock solutions in DMSO (soluble at 200 mg/mL) or ethanol (soluble at 200 mg/mL) for in vitro use; solubility in water is low.  Appearance:  White to off-white powder.  Disposal:  A

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