xcessbio小分子Xcessbio新产品（116）|增长因素（0）|小分子（318）|抗体（37）|
抗体 - **缀合物（8）|即用型套件（5）|文化传媒（0）|肽（0）|当前促销（0）|
定制合成（16）|小型分子库（7）
（+） - JQ1，BET抑制剂
$ 109.00 $ 139.00
目录号 M60139
溴结构域和额外末端（BET）家族蛋白BRD2，BRD3和BRD4的有效和选择性抑制剂
（R）-2-HG，α-KG-依赖性双加氧酶抑制剂 （R）-2-HG，α-KG-依赖性双加氧酶抑制剂
（R）-2-HG，α-KG-依赖性双加氧酶抑制剂
$ 69.00
目录号 M60104
a-KG-依赖性双加氧酶抑制剂
（S）-crizotinib，MTH1抑制剂（S）-crizotinib，MTH1抑制剂
（S）-crizotinib，MTH1抑制剂
$ 99.00
目录号 M60208
一种新型有效的，选择性和细胞渗透性的MTH1抑制剂。
（Z）-4-羟基他莫昔芬，CRISPR编辑增强剂（Z）-4-羟基他莫昔芬，CRISPR编辑增强剂
（Z）-4-羟基他莫昔芬，CRISPR编辑增强剂
$ 89.00
目录号 M60324
以前表征为雌**受体拮抗剂，现在发现可以提高CRISPR介导的基因编辑中的基因组编辑特异性
1,4-DPCA，脯氨酰4-羟化酶（P4H）抑制剂1,4-DPCA，脯氨酰4-羟化酶（P4H）抑制剂
1,4-DPCA，脯氨酰4-羟化酶（P4H）抑制剂
$ 29.00
目录号 M60288
选择性和细胞渗透性脯氨酰4-羟化酶（P4H）抑制剂。
1-甲基-D-色氨酸（D-1MT），IDO抑制剂1-甲基-D-色氨酸（D-1MT），IDO抑制剂
1-甲基-D-色氨酸（D-1MT），IDO抑制剂
$ 29.00
目录号 M60291
一种有效的选择性吲哚胺2,3-双加氧酶（IDO）抑制剂。
4SC-202，HDAC / LSD1双抑制剂 4SC-202，HDAC / LSD1双抑制剂
4SC-202，HDAC / LSD1双抑制剂
$ 109.00
目录号 M60230
一种有效的，选择性和口服生物可用的HDAC / LSD1双重抑制剂。
5-氮杂胞苷，DNA甲基转移酶抑制剂5-氮杂胞苷，DNA甲基转移酶抑制剂
5-氮杂胞苷，DNA甲基转移酶抑制剂
$ 59.00
目录号 M60131
经典的DNA甲基转移酶抑制剂与DNA形成共价加合物，与细胞DNMT结合，消耗酶活性。
A-366，G9a / GLP HMTase抑制剂A-366，G9a / GLP HMTase抑制剂
A-366，G9a / GLP HMTase抑制剂
$ 139.00
目录号 M60210
一种新的高效，选择性和细胞渗透性G9a / GLP组蛋白赖氨酸甲基转移酶抑制剂。
A01，Smurf1 E3泛素连接酶抑制剂A01，Smurf1 E3泛素连接酶抑制剂
A01，Smurf1 E3泛素连接酶抑制剂
$ 109.00
目录号 M60249
一种有效的选择性Smurf1 E3泛素连接酶抑制剂。
A769662，AMPK激动剂A769662，AMPK激动剂
A769662，AMPK激动剂
$ 79.00
目录号 M60020
一种有效的变构AMPK激活剂。
A83-01，TGF-β抑制剂 A83-01，TGF-β抑制剂
A83-01，TGF-β抑制剂
$ 59.00
目录号 M60021
一种有效和选择性的TGF-β途径抑制剂（靶向ALK4，ALK5和ALK7）。
AA92593，黑色素介导的光转导的拮抗剂AA92593，黑色素介导的光转导的拮抗剂
AA92593，黑色素介导的光转导的拮抗剂
$ 139.00
目录号 M60143
黑素蛋白介导的光转导的有效和选择性小分子拮抗剂。
阿比特龙，CYP17抑制剂阿比特龙（CB-7598）阿比特龙，CYP17抑制剂阿比特龙（CB-7598）
阿比特龙，CYP17抑制剂阿比特龙（CB-7598）
$ 69.00
目录号 M60031
首批获得批准用于**去势抵抗性前列腺癌的CYP17抑制剂。
ABT-199，BCL-2抑制剂ABT-199，BCL-2抑制剂
ABT-199，BCL-2抑制剂
$ 99.00
目录号 M60075
一种有效的BCL-2选择性（BCL-X L）抑制剂，具有临床疗效。
ACY-1215（Rocilinostat），HDAC6抑制剂ACY-1215（Rocilinostat），HDAC6抑制剂
ACY-1215（Rocilinostat），HDAC6抑制剂
$ 109.00
目录号 M60076
一种高效，选择性和口服生物可利用的组蛋白脱乙酰酶6（HDAC6）抑制剂。
ADC**单甲基auristatin E（MMAE）ADC**单甲基auristatin E（MMAE）
ADC**单甲基auristatin E（MMAE）
查询
目录号 T60001
用作与抗体连接的**的抗有丝分裂剂。
ADC**单甲基auristatin F（MMAF）ADC**单甲基auristatin F（MMAF）
ADC**单甲基auristatin F（MMAF）
查询
目录号 T60002 xcessbio小分子
用作与抗体连接的**的抗有丝分裂剂
AdipoRon，脂联素受体/ AdipoR激动剂 AdipoRon，脂联素受体/ AdipoR激动剂
AdipoRon，脂联素受体/ AdipoR激动剂
$ 129.00
目录号 M60152
一种新型，高效，选择性和口服活性的脂联素受体小分子激动剂（AdipoR）。
AG-120（Ivosidenib），IDH1抑制剂AG-120（Ivosidenib），IDH1抑制剂
AG-120（Ivosidenib），IDH1抑制剂
$ 129.00
目录号 M60318
临床试验中一种有效，选择性和可逆性IDH1抑制剂。
AG-221（Enasidenib），IHD2抑制剂AG-221（Enasidenib），IHD2抑制剂
AG-221（Enasidenib），IHD2抑制剂
$ 129.00
目录号 M60296
一种有效的选择性IDH2 R140Q突变体抑制剂。
AGI-5198（IDH-C35），突变型IDH1抑制剂 AGI-5198（IDH-C35），突变型IDH1抑制剂
AGI-5198（IDH-C35），突变型IDH1抑制剂
$ 109.00
目录号 M60068
**种高效且选择性的突变体IDH1抑制剂显示在体内具有抗肿瘤效力。
AGI-6780，突变型IDH2抑制剂 AGI-6780，突变型IDH2抑制剂
AGI-6780，突变型IDH2抑制剂
$ 109.00
目录号 M60105
**个高度有效和选择性的小分子突变体IDH2抑制剂。
AK-7，SIRT2抑制剂AK-7，SIRT2抑制剂
AK-7，SIRT2抑制剂
$ 69.00
目录号 M60107
A cell- and brain-permeable, selective sirtuin SIRT2 inhibitor, displays no effect on SIRT1 or SIRT3.
AMI-1，组蛋白甲基转移酶抑制剂AMI-1，组蛋白甲基转移酶抑制剂
AMI-1, Histone Methyltransferase Inhibitor
$79.00
Catalog No. M60272
A potent and specific small molecule inhibitor of histone methyltransferase targeting yeast Hmt1p and human PRMT1.
APY29，IRE1a调制器 APY29，IRE1a调制器
APY29, IRE1a Modulator
$109.00
Catalog No. M60168
A highly potent and selective small molecule modulator of IRE1α.
AR7，RARα拮抗剂 AR7，RARα拮抗剂
AR7, RARα antagonist
$129.00
Catalog No. M60116
A highly potent and selective enhancer of the chaperone-mediated autophagy (CMA) through antagonizing RARα.
AS2034178，GPR40激动剂 AS2034178，GPR40激动剂
AS2034178, GPR40 Agonist
$139.00
Catalog No. M60221
A potent, selective and orally bioavailable GPR40 (FFA1) agonist.
AS8351，KDM5B抑制剂AS8351，KDM5B抑制剂
AS8351, KDM5B Inhibitor
$109.00
Catalog No. M60330
已发现抑制组蛋白去甲基化酶KDM5B（JARID1B）的有效铁螯合剂。
Atglistatin，脂肪甘油三酯脂肪酶（ATGL）抑制剂 Atglistatin，脂肪甘油三酯脂肪酶（ATGL）抑制剂
Atglistatin，脂肪甘油三酯脂肪酶（ATGL）抑制剂
$ 119.00
目录号 M60150
脂肪甘油三酯脂肪酶（ATGL）的高效，选择性和竞争性抑制剂。
AZD2014，mTOR抑制剂AZD2014，mTOR抑制剂
AZD2014，mTOR抑制剂
$ 169.00
目录号 M60090
一种高度有效，选择性和ATP竞争性的mTOR抑制剂，对PIKK家族的其他成员具有高选择性。
AZD6244（塞罗替尼），MEK抑制剂 AZD6244（塞罗替尼），MEK抑制剂
AZD6244（塞罗替尼），MEK抑制剂
$ 109.00
目录号 M60067
临床试验中一种有效且高度选择性的非ATP竞争性MEK抑制剂。
AZD8055，mTOR抑制剂AZD8055，mTOR抑制剂
AZD8055，mTOR抑制剂
$ 69.00
目录号 M60091
一种高度有效，选择性和ATP竞争性mTOR抑制剂，对所有PI3K同种型的选择性> 1,000倍。
叠氮胸苷（AZT），逆转录酶抑制剂 叠氮胸苷（AZT），逆转录酶抑制剂
叠氮胸苷（AZT），逆转录酶抑制剂
$ 29.00
目录号 M60238
一种选择性，口服生物可利用的和脑渗透逆转录酶抑制剂。
b-AP15（NSC687852），去泛素酶抑制剂b-AP15（NSC687852），去泛素酶抑制剂
b-AP15（NSC687852），去泛素酶抑制剂
$ 89.00
目录号 M60251
一种有效的选择性去泛素化酶抑制剂，用于Ub-AMC切割的19S蛋白酶体活性。
BAF312，S1P1 / 5选择性激动剂BAF312，S1P1 / 5选择性激动剂
BAF312，S1P1 / 5选择性激动剂
$ 129.00
目录号 M60039
临床试验中有效和选择性的1-磷酸鞘氨醇（S1P1 / 5）受体激动剂。
BAM7，BAX激活剂BAM7，BAX激活剂
BAM7，BAX激活剂
$ 109.00
目录号 M60069
BAX的**个有效和选择性的小分子激活剂，它是促凋亡BCL-2家族成员。
BAY 87-2243，缺氧诱导因子-1（HIF-1）抑制剂BAY 87-2243，缺氧诱导因子-1（HIF-1）抑制剂
BAY 87-2243，缺氧诱导因子-1（HIF-1）抑制剂
$ 119.00
目录号 M60217
A highly potent and selective hypoxia-inducible factor-1 (HIF-1) inhibitor.
BAY11-7082，E2泛素缀合酶抑制剂BAY11-7082，E2泛素缀合酶抑制剂
BAY11-7082, E2 Ubiquitin Conjugating Enzyme Inhibitor
$89.00
Catalog No. M60309
A potent and selective E2 ubiquitin (Ub) conjugating enzyme inhibitor.
BAZ2-ICR，BAZ2溴结构域抑制剂BAZ2-ICR，BAZ2溴结构域抑制剂
BAZ2-ICR, BAZ2 Bromodomain Inhibitor
$129.00
Catalog No. M60226
A potent and selective BAZ2 bromodomain inhibitor.
BETP，GLP-1R增效剂BETP，GLP-1R增效剂
BETP, GLP-1R Potentiator
$129.00
Catalog No. M60196
A positive allosteric modulator and partial agonist of the glucagon-like peptide 1 (GLP-1) receptor.
BG45，HDAC3抑制剂BG45，HDAC3抑制剂
BG45, HDAC3 Inhibitor
$59.00
Catalog No. M60266
A potent, selective and cell permeable HDAC3 inhibitor.
BI-2536，PLK1和BRD4双重抑制剂 BI-2536，PLK1和BRD4双重抑制剂
BI-2536, PLK1 and BRD4 Dual Inhibitor
$119.00
Catalog No. M60171
BI-2536 is a potent inhibitor of PLK1 (Polo-like kinase 1) and BRD4 in clinical trials.
BI-7273，BRD9溴结构域抑制剂BI-7273，BRD9溴结构域抑制剂
BI-7273, BRD9 Bromodomain Inhibitor
$129.00
Catalog No. M60322
A potent, selective and cell-permeable BRD9 inhibitor.
BI-9564，BRD9溴结构域抑制剂BI-9564，BRD9溴结构域抑制剂
BI-9564, BRD9 Bromodomain Inhibitor
$129.00
Catalog No. M60323
A potent, selective and cell-permeable BRD9 inhibitor.
BIBW2992（阿法替尼），EGFR抑制剂 BIBW2992（阿法替尼），EGFR抑制剂
BIBW2992(Afatinib), EGFR Inhibitor
$109.00
Catalog No. M60065-5s
A potent and selective irreversible inhibitor of EGFR/HER2 in clinical trials.
Bioymifi，TRAIL Receptor DR5 ActivatorBioymifi，TRAIL Receptor DR5 Activator
Bioymifi, TRAIL Receptor DR5 Activator
$109.00
Catalog No. M60088
A potent and selective small molecule agonist of DR5.
BIX-01294，G9a / GLP HMTase抑制剂BIX-01294，G9a / GLP HMTase抑制剂
BIX-01294, G9a/GLP HMTase Inhibitor
$79.00
Catalog No. M60216
A potent and selective G9a and GLP histone lysine methyltransferase inhibitor.
BMI1小鼠单克隆抗体BMI1小鼠单克隆抗体
BMI1 Mouse Monoclonal Antibody
$0.00
Catalog No. A90010-5
BMI1 Mouse Monoclonal Antibody.
BMS-708163（Avagacestat），γ-分泌酶抑制剂BMS-708163（Avagacestat），γ-分泌酶抑制剂
BMS-708163 (Avagacestat), γ-Secretase Inhibitor
$89.00
Catalog No. M60032
A potent γ-secretase Inhibitor, more selective for APP than Notch, in clinical trials for Alzheimer's disease.
BQU57，GTP酶Ral抑制剂BQU57，GTP酶Ral抑制剂
BQU57, GTPase Ral Inhibitor
$139.00
Catalog No. M60228
A potent and selective GTPase Ral Inhibitor
BRD9757，HDAC6抑制剂BRD9757，HDAC6抑制剂
BRD9757, HDAC6 Inhibitor
$129.00
Catalog No. M60117
A highly potent and selective HDAC6 inhibitor.
溴代***，泛溴代域抑制剂溴代***，泛溴代域抑制剂
Bromosporine, Pan-bromodomain Inhibitor
$129.00
Catalog No. M60144
A broad spectrum inhibitor for bromodomains.
C646，p300 / CBP抑制剂C646，p300 / CBP抑制剂
C646, p300/CBP inhibitor
$129.00
Catalog No. M60129
A potent, selective and cell-permeable p300/CBP histone acetyltransferase (HAT) inhibitor.
Carfilzomib，蛋白酶体抑制剂Carfilzomib，蛋白酶体抑制剂
Carfilzomib, Proteasome Inhibitor
$109.00
Catalog No. M60109
A selective, irreversible proteasome inhibitor.
CASIN，Cdc42抑制剂 CASIN，Cdc42抑制剂
CASIN，Cdc42抑制剂
$ 139.00
目录号 M60040
一种新的有效的Cdc42抑制剂; 被证明可以挽救HSC衰老表型并促进HSC移植效率。
CAY10603，HDAC6抑制剂CAY10603，HDAC6抑制剂
CAY10603，HDAC6抑制剂
$ 129.00
目录号 M60234
一种有效的选择性HDAC6抑制剂。
CB-5083，p97 AAA ATPase抑制剂 CB-5083，p97 AAA ATPase抑制剂
CB-5083，p97 AAA ATPase抑制剂
$ 129.00
目录号 M60306
一种高效，选择性和口服生物可利用的p97 AAA ATP酶抑制剂。
CBX5多克隆抗体CBX5多克隆抗体
CBX5多克隆抗体
$ 0.00包装
目录号 A70033
Chromobox蛋白同系物5
CHIR99021，GSK3β抑制剂 CHIR99021，GSK3β抑制剂
CHIR99021，GSK3β抑制剂
$ 390.00
目录号 M60002
*广泛使用的，有效的和选择性的GSK3β抑制剂; Wnt通路激活剂。
CI994（Tacedinaline），HDAC抑制剂CI994（Tacedinaline），HDAC抑制剂
CI994（Tacedinaline），HDAC抑制剂
$ 59.00
目录号 M60186
一种有效的，选择性和口服有效的靶向HDAC1，HDAC2和HDAC3的组蛋白去乙酰化酶（HDAC）抑制剂。
Cilliobrevin D，AAA + ATPase运动细胞质动力蛋白抑制剂 Cilliobrevin D，AAA + ATPase运动细胞质动力蛋白抑制剂
Cilliobrevin D，AAA + ATPase运动细胞质动力蛋白抑制剂
$ 139.00
目录号 M60041-2s
AAA + ATPase运动细胞质动力蛋白的新型和特异性抑制剂; 扰乱主要纤毛内的蛋白质运输并且影响其他动力依赖过程，例如培养细胞中的纺锤体极点聚焦，动粒 - 微管附着，黑素体聚集和过氧化物酶体动力。
Bromodomain / BET化合物库Bromodomain / BET化合物库
Bromodomain / BET化合物库
$ 1150.00 $ 1437.00
目录号 LI30006
溴代域/ BET组化合物文库由分开的小瓶中的23个小分子组成。
HDAC的化合物库HDAC的化合物库
HDAC的化合物库
$ 700.00 $ 850.00
目录号 LI30005
Compound Library of HDAC set is composed of 18 small molecules in separated vials.
组蛋白去甲基化酶复合文库组蛋白去甲基化酶复合文库
Compound Library of Histone Demethylase
$1400.00
Catalog No. LI30003
Library of Histone Demethylase is composed of 15 small molecules in separated vials.
组蛋白甲基转移酶复合文库组蛋白甲基转移酶复合文库
Compound Library of Histone Methyltransferase
$1200.00
Catalog No. LI30002
Compound Library of Histone Methyltransferase is composed of 14 small molecules in separated vials.
缺氧诱导因子化合物库缺氧诱导因子化合物库
Compound Library of Hypoxia Inducible Factor
$360.00 $446.00
Catalog No. LI30007
Epigenetic compounds library of Hypoxia Inducible Factor
CP-690550，JAK抑制剂CP-690550，JAK抑制剂
CP-690550, JAK Inhibitor
$79.00
Catalog No. M60033
A potent and selective pan-JAK Inhibitor in clinical trials for rheumatoid arthritis.
CPI-169，EZH2甲基转移酶抑制剂CPI-169，EZH2甲基转移酶抑制剂
CPI-169, EZH2 Methyltransferase Inhibitor
$129.00
目录号 M60275
组蛋白甲基转移酶EZH2的高效和选择性小分子抑制剂。
CPI-455，KDM5脱甲基酶抑制剂 CPI-455，KDM5脱甲基酶抑制剂
CPI-455，KDM5脱甲基酶抑制剂
$ 129.00
目录号 M60326
一种有效的选择性KDM5A抑制剂。
CPI203，BET抑制剂CPI203，BET抑制剂
CPI203，BET抑制剂
$ 139.00
目录号 M60124
一种新的有效的，选择性的和细胞渗透性的溴结构域和额外终端（BET）家族蛋白BRD4的抑制剂，抑制Myc表达。
CRISPR编辑工具箱CRISPR编辑工具箱
CRISPR编辑工具箱
$ 499.00
目录号 LI30010
CRISPR编辑的复合集合。
CTEP，mGlu5拮抗剂CTEP，mGlu5拮抗剂
CTEP，mGlu5拮抗剂
$ 259.00
目录号 M60099
mGlu5受体的高效，选择性和口服生物可利用的变构拮抗剂。
CUDC-101，HDAC / EGFR / HER2抑制剂 CUDC-101，HDAC / EGFR / HER2抑制剂
CUDC-101，HDAC / EGFR / HER2抑制剂
$ 69.00
目录号 M60092
在临床试验中靶向HDAC，EGFR和HER2的强效多靶点抑制剂。
CUDC-907，PI3K / HDAC双重抑制剂CUDC-907，PI3K / HDAC双重抑制剂
CUDC-907，PI3K / HDAC双重抑制剂
$ 139.00
目录号 M60077
临床试验中一种强效的I类PI3K激酶和HDAC的双重抑制剂。
定制合成产品1定制合成产品1
定制合成产品1
$ 5000.00
目录号 CS-1
CX-4945，CK2（酪蛋白激酶2）抑制剂CX-4945，CK2（酪蛋白激酶2）抑制剂
CX-4945，CK2（酪蛋白激酶2）抑制剂
$ 129.00
目录号 M60267
一种有效的，选择性和生物可利用的CK2（酪蛋白激酶2）抑制剂。
CX-5461，RNA聚合酶I抑制剂CX-5461，RNA聚合酶I抑制剂
CX-5461，RNA聚合酶I抑制剂
$ 149.00
目录号 M66052
一种有效的选择性RNA聚合酶I抑制剂，用于抗肿瘤应用。
环杷明，刺猬拮抗剂环杷明，刺猬拮抗剂
环杷明，刺猬拮抗剂
$ 79.00
目录号 M60022
刺猬拮抗剂的强效天然产物; 直接绑定到Smoothened / Smo。
环孢菌素A，MPTP抑制剂和HSC保护剂环孢菌素A，MPTP抑制剂和HSC保护剂
环孢菌素A，MPTP抑制剂和HSC保护剂
$ 39.00
Catalog No. M60262
An inhibitor of the mitochondrial permeability transition pore (MPTP).
大豆苷元-2c，成骨调节剂大豆苷元-2c，成骨调节剂
Daidzein-2c, Osteogenic Modulator
$109.00
Catalog No. M60158
A potent synthetic daidzein analog with osteogenic induction potentials on human Mesenchymal Stem Cells (MSC).
Daminozide --- KDM2 / 7组蛋白脱甲基酶抑制剂Daminozide --- KDM2 / 7组蛋白脱甲基酶抑制剂
Daminozide --- KDM2/7 Histone Demethylases Inhibitor
$69.00
Catalog No. M60074
A potent and selective small molecule inhibitor of the KDM2/7 family of human JmjC histone demethylases.
DAPT，γ-分泌酶抑制剂DAPT，γ-分泌酶抑制剂
DAPT, γ-secretase Inhibitor
$300.00
Catalog No. M60023
A γ-secretase inhibitor and widely used as a Notch pathway inhibitor.
DASA-58（ML203），丙酮酸激酶M2（PKM2）激活剂DASA-58（ML203），丙酮酸激酶M2（PKM2）激活剂
DASA-58 (ML203), Pyruvate Kinase M2 (PKM2) Activator
$109.00
Catalog No. M60305
A potent and selective Pyruvate kinase M2 (PKM2) activator.
Deltarasin，KRAS-PDEδ抑制剂Deltarasin，KRAS-PDEδ抑制剂
Deltarasin, KRAS-PDEδ Inhibitor
$139.00
目录号 M60218
KRAS-PDEδ相互作用的有效和选择性小分子抑制剂
演示演示
演示
$ 0.00包装
目录号 123456
DMOG，脯氨酰4-羟化酶（P4H）抑制剂DMOG，脯氨酰4-羟化酶（P4H）抑制剂
DMOG，脯氨酰4-羟化酶（P4H）抑制剂
$ 39.00
目录号 M60287
选择性，竞争性和细胞渗透性脯氨酰4-羟化酶（P4H）抑制剂。
DMXAA（Vadimezan），mSTING激动剂DMXAA（Vadimezan），mSTING激动剂
DMXAA（Vadimezan），mSTING激动剂
$ 79.00
目录号 M60301
一种有效和选择性的mSTING激动剂，对STING的选择性小于STING。
DNMT3A多克隆抗体DNMT3A多克隆抗体
DNMT3A多克隆抗体
$ 0.00包装
目录号 A70035
DNA（胞嘧啶-5）甲基转移酶3A（DNMT3A）
DZNep（3-Deazaneplanocin A）---组蛋白甲基转移酶抑制剂 DZNep（3-Deazaneplanocin A）---组蛋白甲基转移酶抑制剂
DZNep（3-Deazaneplanocin A）---组蛋白甲基转移酶抑制剂
$ 129.00
目录号 M60141
一种S-腺苷高半胱氨酸水解酶抑制剂，间接抑制组蛋白甲基转移酶并降低全局DNA甲基化
EED226，PRC2抑制剂EED226，PRC2抑制剂
EED226，PRC2抑制剂
$ 139.00
目录号 M60327
直接与EED的H3K27me3结合口袋结合的强效和选择性变构PRC2抑制剂。
EML425，CBP / p300抑制剂EML425，CBP / p300抑制剂
EML425，CBP / p300抑制剂
$ 129.00
目录号 M60257
选择性，非竞争性和细胞渗透性KAT3组蛋白乙酰转移酶CBP / p300抑制剂。
Entinostat（MS-275）-HDAC抑制剂 Entinostat（MS-275）-HDAC抑制剂
Entinostat（MS-275）-HDAC抑制剂
$ 59.00
目录号 M60174
Entinostat（MS-275）是一种有效的选择性HDAC1和HDAC3抑制剂。
EPZ-5676 --- DOT1L抑制剂EPZ-5676 --- DOT1L抑制剂
EPZ-5676 --- DOT1L抑制剂
$ 139.00
目录号 M60123
DOT1L甲基转移酶的高度有效和选择性抑制剂，Ki为70 pM，选择性阻断辅因子S-腺苷甲硫氨酸的结合。
EPZ-6438，EZH2甲基转移酶抑制剂EPZ-6438，EZH2甲基转移酶抑制剂
EPZ-6438，EZH2甲基转移酶抑制剂
$ 129.00
目录号 M60122
EPZ-6438（E7438）是一种有效的选择性小分子组蛋白甲基转移酶EZH2的小分子抑制剂，用于临床开发。
EPZ015666（GSK3235025），PRMT5抑制剂 EPZ015666（GSK3235025），PRMT5抑制剂
EPZ015666（GSK3235025），PRMT5抑制剂
$ 129.00
目录号 M60254
一种有效的，选择性和口服生物可利用的蛋白精氨酸甲基转移酶-5（PRMT5）抑制剂。
EX-527，SIRT1抑制剂EX-527，SIRT1抑制剂
EX-527，SIRT1抑制剂
$ 69.00
目录号 M60108
EX-527是一种高度有效的选择性SIRT1抑制剂，IC50〜98 nM。
EZH2 Polyclonal AntibodyEZH2 Polyclonal Antibody
EZH2多克隆抗体
$ 0.00包装
目录号 A70036
组蛋白 - 赖氨酸N-甲基转移酶EZH2
FASCIN-G2, Fascin InhibitorFASCIN-G2, Fascin Inhibitor
FASCIN-G2，Fascin抑制剂
$ 129.00
目录号 M60269
一种有效的，选择性和生物可利用的小分子，可抑制肌成束蛋白的肌动蛋白捆绑活性。
Fatostatin A, Sterol Regulatory Binding Proteins (SREBPs) InhibitorFatostatin A, Sterol Regulatory Binding Proteins (SREBPs) Inhibitor
脂肪抑制素A，固醇调节性结合蛋白（SREBPs）抑制剂
$ 59.00
目录号 M60180
Fatostatin A is a highly potent, specific and cell permeable inhibitor of Sterol Regulatory Binding Proteins (SREBPs).
Ferrostatin-1 (Fer-1), Ferroptosis Inhibitor Ferrostatin-1 (Fer-1), Ferroptosis Inhibitor
Ferrostatin-1 (Fer-1), Ferroptosis Inhibitor
$109.00
Catalog No. M60042
Ferrostatin-1 (Fer-1) is a potent inhibitor of ferroptosis with an EC50 ~60 nM, identified by a HTS using erastin-induced ferroptosis in HT-1080 cells.
FG-4592 (Roxadustat), HIF Prolyl-Hydroxylases InhibitorFG-4592 (Roxadustat), HIF Prolyl-Hydroxylases Inhibitor
FG-4592 (Roxadustat), HIF Prolyl-Hydroxylases Inhibitor
$39.00
Catalog No. M60263
A potent, selective and bioavailable inhibitor of hypoxia-inducible factor prolyl hydroxylase.
FH1, Hepatocytes Functional EnhancerFH1, Hepatocytes Functional Enhancer
FH1, Hepatocytes Functional Enhancer
$139.00
Catalog No. M60127
FH1 is a potent and selective small molecule that enhances hepatocyte functions and promotes the differentiation and maturation of iPSC-derived hepatocytes toward a more mature phenotype in vitro.
FLI-06, Notch Pathway ModulatorFLI-06, Notch Pathway Modulator
FLI-06, Notch Pathway Modulator
$139.00
Catalog No. M60149
FLI-06 is a novel potent and selective small molecule intercepting Notch signaling and the early secretory pathway (EC50 ~2.3 µM), identified by using automated microscopy to monitor the trafficking and processing of a ligand-independent Notch-GFP fusion reporter.
Fmoc-Ala-Ala-Asn-PAB-PNPFmoc-Ala-Ala-Asn-PAB-PNP
Fmoc-Ala-Ala-Asn-PAB-PNP
Inquiry
Catalog No. L60002
Peptide prodrug linker
Fmoc-Val-Cit-PABFmoc-Val-Cit-PAB
Fmoc-Val-Cit-PAB
Inquiry
Catalog No. L60001
Peptide prodrug linker
Forskolin, Adenylyl Cyclase Activator Forskolin, Adenylyl Cyclase Activator
Forskolin, Adenylyl Cyclase Activator
$79.00
Catalog No. M60024 xcessbio小分子
A potent adenylate cyclase activator to increase the intracellular levels of cAMP.
FPH1, Hepatocytes Functional Proliferation InducerFPH1, Hepatocytes Functional Proliferation Inducer
FPH1, Hepatocytes Functional Proliferation Inducer
$139.00
Catalog No. M60126
FPH1 is a potent and selective small molecule that induced Functional Proliferation of primary human Hepatocytes in vitro, identified by a high-throughput, cell-based screening using primary human hepatocytes.
Furamidine, PRMT1 InhibitorFuramidine, PRMT1 Inhibitor
Furamidine, PRMT1 Inhibitor
$99.00
Catalog No. M60256
A potent, selective and cell permeable Protein arginine methyltransferase-1 (PRMT1) inhibitor.
GDC-0068, Akt Inhibitor GDC-0068, Akt Inhibitor
GDC-0068, Akt Inhibitor
$159.00
Catalog No. M60066
A novel potent and selective ATP competitive Akt inhibitor in clinical trials.
GDC-0349, mTOR Inhibitor GDC-0349, mTOR Inhibitor
GDC-0349, mTOR Inhibitor
$129.00
Catalog No. M60110
A potent and selective ATP-competitive inhibitor of mTOR in clinical trials.
GDC-0449 (Vismodegib), Hedgehog Antagonist GDC-0449 (Vismodegib), Hedgehog Antagonist
GDC-0449 (Vismodegib), Hedgehog Antagonist
$79.00
Catalog No. M60034
A potent and specific hedgehog pathway inhibitor approved by FDA
GDC-0941, PI3K Inhibitor GDC-0941, PI3K Inhibitor
GDC-0941, PI3K Inhibitor
$79.00
Catalog No. M60111
A highly potent, selective and orally bioavailable class-I PI3K kinase inhibitor.
GN44028, HIF-1α InhibitorGN44028, HIF-1α Inhibitor
GN44028, HIF-1α Inhibitor
$89.00
Catalog No. M60325
A potent and selective HIF-1α inhibitor.
GNF-7, Ras Signaling InhibitorGNF-7, Ras Signaling Inhibitor
GNF-7, Ras Signaling Inhibitor
$129.00
Catalog No. M60281
A potent, selective and bioavailable Ras signaling inhibitor.
GNF4877, β Cell Proliferation Inducer GNF4877, β Cell Proliferation Inducer
GNF4877, β Cell Proliferation Inducer
$159.00
Catalog No. M60294
A highly potent and selective small molecule that promotes pancreatic β cell proliferation in rodent and human primary islets.
GNF7156, β Cell Proliferation Inducer GNF7156, β Cell Proliferation Inducer
GNF7156, β Cell Proliferation Inducer
$139.00
Catalog No. M60293
A highly potent and selective small molecule that promotes pancreatic β cell proliferation in rodent and human primary islets.
Go6893, PKC InhibitorGo6893, PKC Inhibitor
Go6893, PKC Inhibitor
$129.00
Catalog No. M60273
A potent pan-PKC inhibitor.
GPR39-C3, GPR39 AgonistGPR39-C3, GPR39 Agonist
GPR39-C3, GPR39 Agonist
$139.00
Catalog No. M60209
The first potent, selective and orally bioavailable GPR39 agonist.
GPR39-C3bulkGPR39-C3bulk
GPR39-C3bulk
$0.00 $875.00
Catalog No. M60209-b
GS143, IkappaB Ubiquitination Inhibitor GS143, IkappaB Ubiquitination Inhibitor
GS143, IkappaB Ubiquitination Inhibitor
$129.00
Catalog No. M60308
A selective β-TrCP1 ligase inhibitor
GSK-J1, H3K27 Histone Demethylases UTX and JMJD3 Inhibitor GSK-J1, H3K27 Histone Demethylases UTX and JMJD3 Inhibitor
GSK-J1, H3K27 Histone Demethylases UTX and JMJD3 Inhibitor
$109.00
Catalog No. M60062
The first selective and potent inhibitor of the H3K27 histone demethylases UTX and JMJD3.
GSK-J4，H3K27组蛋白脱甲基酶UTX和JMJD3抑制剂 GSK-J4，H3K27组蛋白脱甲基酶UTX和JMJD3抑制剂
GSK-J4, H3K27 Histone Demethylases UTX and JMJD3 Inhibitor
$109.00
Catalog No. M60063
An ethyl ester derivative of GSK-J1 as a pro-drug for cellular assays; the first selective and potent inhibitor of the H3K27 histone demethylases UTX and JMJD3.
GSK-J4bulkGSK-J4bulk
GSK-J4bulk
$0.00
Catalog No. M60063-b
GSK-LSD1，LSD1抑制剂GSK-LSD1，LSD1抑制剂
GSK-LSD1, LSD1 Inhibitor
$139.00
Catalog No. M60179
赖氨酸特异性去甲基化酶-1（LSD1）的高度有效，特异性和不可逆转抑制剂。
GSK126，EZH2甲基转移酶抑制剂。GSK126，EZH2甲基转移酶抑制剂。
GSK126，EZH2甲基转移酶抑制剂。
$ 129.00
目录号 M60071
GSK126是一种高效且具有选择性的组蛋白甲基转移酶EZH2的小分子抑制剂。
GSK126bulkGSK126bulk
GSK126bulk
$ 0.00包装
目录号 M60071-b
GSK2801，Bromodomain BAZ2A / B抑制剂GSK2801，Bromodomain BAZ2A / B抑制剂
GSK2801，Bromodomain BAZ2A / B抑制剂
$ 129.00
目录号 M60283
溴结构域BAZ2A和BAZ2B的有效，选择性和细胞渗透性抑制剂。
GSK2879552，LSD1抑制剂GSK2879552，LSD1抑制剂
GSK2879552，LSD1抑制剂
$ 129.00
目录号 M60297
赖氨酸特异性脱甲基酶1（LSD1）的高效，选择性和口服生物可利用的不可逆抑制剂。
GSK343，EZH2甲基转移酶抑制剂GSK343，EZH2甲基转移酶抑制剂
GSK343，EZH2甲基转移酶抑制剂
$ 79.00
目录号 M60173
GSK343是一种有效的选择性组蛋白甲基转移酶EZH2的小分子抑制剂。
GSK591（EPZ015866），PRMT5抑制剂GSK591（EPZ015866），PRMT5抑制剂
GSK591（EPZ015866），PRMT5抑制剂
$ 109.00
目录号 M60321
一种有效和选择性蛋白精氨酸甲基转移酶-5（PRMT5）抑制剂。
GSK5959，BRPF1溴结构域抑制剂GSK5959，BRPF1溴结构域抑制剂
GSK5959，BRPF1溴结构域抑制剂
$ 129.00
目录号 M60239
一种有效的，选择性和细胞渗透性的BRPF1溴结构域抑制剂。
H3K36me3小鼠单克隆抗体H3K36me3小鼠单克隆抗体
H3K36me3小鼠单克隆抗体
$ 0.00包装
目录号 A90004
H3K36me3小鼠单克隆抗体
H3K4me1多克隆抗体H3K4me1多克隆抗体
H3K4me1多克隆抗体
查询
目录号 A70010
单甲基化的H3K4多克隆抗体
H3K4me3小鼠单克隆抗体H3K4me3小鼠单克隆抗体
H3K4me3小鼠单克隆抗体
查询
目录号 A90006
H3K4me3小鼠单克隆抗体
H3K79me1小鼠单克隆抗体H3K79me1小鼠单克隆抗体
H3K79me1小鼠单克隆抗体
查询
目录号 A90001
H3K79me1小鼠单克隆抗体
H3K79me2小鼠单克隆抗体H3K79me2小鼠单克隆抗体
H3K79me2小鼠单克隆抗体
查询
目录号 A90002
H3K79me2小鼠单克隆抗体
H3K79me3小鼠单克隆抗体H3K79me3小鼠单克隆抗体
H3K79me3 Mouse Monoclonal Antibody
Inquiry
Catalog No. A90003
H3K79me3 Mouse Monoclonal Antibody
H3K9（Ac）K14（Ac）兔pAbH3K9（Ac）K14（Ac）兔pAb
H3K9(Ac)K14(Ac) Rabbit pAb
$250.00
Catalog No. A-10001-100
H3K9me3小鼠单克隆抗体H3K9me3小鼠单克隆抗体
H3K9me3 Mouse Monoclonal Antibody
Inquiry
Catalog No. A90005
H3K9me3 Mouse Monoclonal Antibody
Harmine，DYRK1A抑制剂Harmine，DYRK1A抑制剂
Harmine, DYRK1A Inhibitor
$29.00
Catalog No. M60241
A potent, selective and orally bioavailable DYRK1A inhibitor.
HBX41108，USP7抑制剂HBX41108，USP7抑制剂
HBX41108, USP7 Inhibitor
$129.00
Catalog No. M60244
A potent and selective ubiquitin-specific protease 7 (USP7) inhibitor.
HCI-2509（SP2509），可逆LSD1抑制剂。HCI-2509（SP2509），可逆LSD1抑制剂。
HCI-2509 (SP2509), Reversible LSD1 Inhibitor.
$109.00
Catalog No. M60160
A highly potent, specific, and reversible Lysine Specific Demethylase-1 (LSD1) inhibitor with in vivo efficacy.
HDAC4小鼠单克隆抗体HDAC4小鼠单克隆抗体
HDAC4 Mouse Monoclonal Antibody
Inquiry
Catalog No. A90011
组蛋白去乙酰化酶4（HDAC4）是一种组蛋白脱乙酰酶，其在连接到启动子时抑制转录。
HDAC4多克隆抗体HDAC4多克隆抗体
HDAC4多克隆抗体
查询
目录号 A70037
组蛋白脱乙酰酶4
Heclin，HECT E3泛素连接酶抑制剂Heclin，HECT E3泛素连接酶抑制剂
Heclin，HECT E3泛素连接酶抑制剂
$ 89.00
目录号 M60248
选择性HECT E3泛素连接酶抑制剂抑制Nedd4，Smurf2和WWP1。
HG-10-102-01，LRRK2抑制剂 HG-10-102-01，LRRK2抑制剂
HG-10-102-01，LRRK2抑制剂
$ 139.00
目录号 M60061
野生型LRRK2和G2019S突变体的脑渗透剂有效和选择性抑制剂。
Hh-Ag1.5，刺猬激动剂 Hh-Ag1.5，刺猬激动剂
Hh-Ag1.5，刺猬激动剂
$ 139.00
目录号 M60004
Hh通路中*有效和选择性的激动剂（Smoothened / Smo激动剂）; 可以取代重组Hh蛋白以激活Hh途径
HIF-C2，HIF-2抑制剂 HIF-C2，HIF-2抑制剂
HIF-C2，HIF-2抑制剂
$ 139.00
目录号 M60121
缺氧诱导因子-2（HIF-2）的有效选择性变构抑制剂。
组蛋白H3K27me1多克隆抗体组蛋白H3K27me1多克隆抗体
组蛋白H3K27me1多克隆抗体
查询
目录号 A70013
含有单甲基赖氨酸27的组蛋白H3
组蛋白H3K27me2多克隆抗体组蛋白H3K27me2多克隆抗体
组蛋白H3K27me2多克隆抗体
查询
目录号 A70014
含有二甲基化赖氨酸的组蛋白H3 27
组蛋白H3K27me3多克隆抗体组蛋白H3K27me3多克隆抗体
组蛋白H3K27me3多克隆抗体
查询
目录号 A70015
含有**基赖氨酸27的组蛋白H3
组蛋白H3K36me1多克隆抗体组蛋白H3K36me1多克隆抗体
组蛋白H3K36me1多克隆抗体
查询
目录号 A70016
含有单甲基化赖氨酸的组蛋白H3 36
组蛋白H3K36me2多克隆抗体组蛋白H3K36me2多克隆抗体
组蛋白H3K36me2多克隆抗体
查询
目录号 A70017
含有二甲基化赖氨酸的组蛋白H3 36
组蛋白H3K36me3多克隆抗体组蛋白H3K36me3多克隆抗体
组蛋白H3K36me3多克隆抗体
查询
目录号 A70018
含有**基赖氨酸的组蛋白H3 36
组蛋白H3K4me2多克隆抗体组蛋白H3K4me2多克隆抗体
组蛋白H3K4me2多克隆抗体
查询
目录号 A70011
含有二甲基赖氨酸的组蛋白H3 4
组蛋白H3K4me3多克隆抗体组蛋白H3K4me3多克隆抗体
组蛋白H3K4me3多克隆抗体
查询
目录号 A70012
含有**基赖氨酸的组蛋白H3 4
组蛋白H3K79me1多克隆抗体组蛋白H3K79me1多克隆抗体
组蛋白H3K79me1多克隆抗体
查询
目录号 A70019
含有单甲基化赖氨酸79的组蛋白H3
组蛋白H3K79me2多克隆抗体组蛋白H3K79me2多克隆抗体
组蛋白H3K79me2多克隆抗体
查询
目录号 A70020
含有二甲基赖氨酸79的组蛋白H3
组蛋白H3K79me3多克隆抗体组蛋白H3K79me3多克隆抗体
组蛋白H3K79me3多克隆抗体
查询
目录号 A70021
含有**基赖氨酸79的组蛋白H3
组蛋白H3K9me1多克隆抗体组蛋白H3K9me1多克隆抗体
组蛋白H3K9me1多克隆抗体
查询
目录号 A70022
含有单甲基赖氨酸9的组蛋白H3
组蛋白H3K9me2多克隆抗体组蛋白H3K9me2多克隆抗体
组蛋白H3K9me2多克隆抗体
查询
目录号 A70023
histone H3 containing the dimethylated lysine 9
组蛋白H3K9me3多克隆抗体组蛋白H3K9me3多克隆抗体
Histone H3K9me3 Polyclonal Antibody
Inquiry
Catalog No. A70024
histone H3 containing the trimethylated lysine 9
组蛋白H3R26me1多克隆抗体组蛋白H3R26me1多克隆抗体
Histone H3R26me1 Polyclonal Antibody
Inquiry
Catalog No. A70031
histone H3 containing the monomethylated Arg26
组蛋白H3R26me2a多克隆抗体组蛋白H3R26me2a多克隆抗体
Histone H3R26me2a Polyclonal Antibody
Inquiry
Catalog No. A70032
histone H3 containing the asymmetrically dimethylated Arg26
组蛋白H3R2me1多克隆抗体组蛋白H3R2me1多克隆抗体
Histone H3R2me1 Polyclonal Antibody
Inquiry
Catalog No. A70029
histone H3 containing the monomethylated Arg2
组蛋白H3R2me2a多克隆抗体组蛋白H3R2me2a多克隆抗体
Histone H3R2me2a Polyclonal Antibody
Inquiry
Catalog No. A70028
histone H3 containing the asymmetrically dimethylated Arg2
组蛋白H3R2me2s多克隆抗体组蛋白H3R2me2s多克隆抗体
Histone H3R2me2s Polyclonal Antibody
Inquiry
Catalog No. A70030
histone H3 containing the symmetrically dimethylated Arg2
组蛋白H4R3me1多克隆抗体组蛋白H4R3me1多克隆抗体
Histone H4R3me1 Polyclonal Antibody
Inquiry
Catalog No. A70025
histone H4 containing the monomethylated Arg3
组蛋白H4R3me2a多克隆抗体组蛋白H4R3me2a多克隆抗体
Histone H4R3me2a Polyclonal Antibody
Inquiry
Catalog No. A70027
histone H4 containing the asymmetrically dimethylated Arg3
组蛋白H4R3me2s多克隆抗体组蛋白H4R3me2s多克隆抗体
Histone H4R3me2s Polyclonal Antibody
Inquiry
Catalog No. A70026
histone H4 containing the symmetrically dimethylated Arg3
HLCL-61，PRMT5抑制剂HLCL-61，PRMT5抑制剂
HLCL-61, PRMT5 Inhibitor
$109.00
Catalog No. M60320
A potent and selective Protein arginine methyltransferase-5 (PRMT5) Inhibitor.
HLY78，Wnt激动剂HLY78，Wnt激动剂
HLY78, Wnt Activator
$149.00
Catalog No. M60140
An activator of the Wnt pathway by targeting the DIX domain of Axin and potentiating the Axin–LRP6 association, thus promoting LRP6 phosphorylation and Wnt signaling transduction.
HPOB，HDAC6抑制剂HPOB，HDAC6抑制剂
HPOB, HDAC6 Inhibitor
$79.00
Catalog No. M60231
A potent and selective HDAC6 inhibitor.
Hydroxychloroquine (HCQ), Autophagy and TLR9 Inhibitor Hydroxychloroquine (HCQ), Autophagy and TLR9 Inhibitor
Hydroxychloroquine (HCQ), Autophagy and TLR9 Inhibitor
$49.00
Catalog No. M60302
A potent autophagy inhibitor and TLR9 inhibitor
I-BET151 (GSK1210151A), BET Inhibitor I-BET151 (GSK1210151A), BET Inhibitor
I-BET151 (GSK1210151A), BET Inhibitor
$109.00
Catalog No. M66053
A potent and selective inhibitor of the bromodomain and extra terminal (BET) family proteins BRD2, BRD3, and BRD4.
I-BET762 (GSK525762), BET Inhibitor I-BET762 (GSK525762), BET Inhibitor
I-BET762 (GSK525762), BET Inhibitor
$139.00
Catalog No. M60154
A novel, highly potent, selective and cell permeable BET inhibitor in clinical trials.
I-BRD9, Bromodomain Containing Protein 9 (BRD9) InhibitorI-BRD9, Bromodomain Containing Protein 9 (BRD9) Inhibitor
I-BRD9, Bromodomain Containing Protein 9 (BRD9) Inhibitor
$129.00
Catalog No. M60276
A potent, selective and cell permeable Bromodomain Containing Protein 9 (BRD9) inhibitor.
I-CBP112, p300/CBP Bromodomain Inhibitor I-CBP112, p300/CBP Bromodomain Inhibitor
I-CBP112, p300/CBP Bromodomain Inhibitor
$139.00
Catalog No. M60128
A highly potent and selective p300/CBP bromodomain inhibitor.
ID-8, DYRK InhibitorID-8, DYRK Inhibitor
ID-8, DYRK Inhibitor
$89.00
Catalog No. M60102
A potent and selective small molecule inhibitor of dual-specificity tyrosine phosphorylation- regulated kinase (DYRK).
IDH-C227, IDH1 Inhibitor IDH-C227, IDH1 Inhibitor
IDH-C227, IDH1 Inhibitor
$139.00
Catalog No. M60043
A potent and selective inhibitor of the IDH1 R132H mutant with good cellular activity.
IDH2-C100, IHD2 Inhibitor IDH2-C100, IHD2 Inhibitor
IDH2-C100, IHD2 Inhibitor
$129.00
Catalog No. M60190
A potent and selective inhibitor of IDH2 R140Q and R172K mutant.
IDH2-C100BulkIDH2-C100Bulk
IDH2-C100Bulk
$750.00 $990.00
Catalog No. M60190-b
iN-LSCiN-LSC
iN-LSC
$89.00
Catalog No. S10004
Combination of LDN193189 (BMP inhibitor), SB431542 (TGFβ inhibitor), and CHIR99021 (GSK3 inhibitor) can enhance reprogramming of human fibroblasts into induced neurons.
INCB024360 (Epacadostat), IDO InhibitorINCB024360 (Epacadostat), IDO Inhibitor
INCB024360 (Epacadostat), IDO Inhibitor
$109.00
Catalog No. M60292
A potent and selective indoleamine 2,3-dioxygenase (IDO1) inhibitor.
INDY, DYRK1A/B InhibitorINDY, DYRK1A/B Inhibitor
INDY, DYRK1A/B Inhibitor
$79.00
Catalog No. M60242
A potent and selective DYRK1A/B inhibitor.
IOX1, 2OG Oxygenases InhibitorIOX1, 2OG Oxygenases Inhibitor
IOX1, 2OG Oxygenases Inhibitor
$109.00
Catalog No. M60195
A cell-permeable broad-spectrum inhibitor of most 2OG oxygenases.
IOX2, HIF Prolyl-Hydroxylases (PHD2) Inhibitor IOX2, HIF Prolyl-Hydroxylases (PHD2) Inhibitor
IOX2, HIF Prolyl-Hydroxylases (PHD2) Inhibitor
$89.00
Catalog No. M66054
A potent and selective PHD (HIF prolyl-hydroxylases) inhibitor with cellular activity.
IOX4, PHD2 InhibitorIOX4, PHD2 Inhibitor
IOX4, PHD2 Inhibitor
$109.00
Catalog No. M60284
A potent and selective PHD2 inhibitor.
iPSC-TSPCiPSC-TSPC
iPSC-TSPC
$109.00
Catalog No. S10005
Combination of Thiazovivin (ROCK inhibitor), SB431542 (TGFβ inhibitor), PD0325901 (MEK inhibitor), and CHIR99021 (GSK3 inhibitor) can enhance and accelerate reprogramming of human somatic cells (e.g., fibroblasts) into iPSCs.
IRE-3, IRE1a Modulator IRE-3, IRE1a Modulator
IRE-3, IRE1a Modulator
$129.00
Catalog No. M60167
A highly potent and selective small molecule modulator of IRE1α.
Ischemin, CBP Bromodomain Inhibitor Ischemin, CBP Bromodomain Inhibitor
Ischemin, CBP Bromodomain Inhibitor
$79.00
Catalog No. M60229
A potent, selective and cell permeable CBP bromodomain inhibitor.
ISRIB (trans-isomer), Inhibitor of “Integrated Stress Response” (ISR)ISRIB (trans-isomer), Inhibitor of “Integrated Stress Response” (ISR)
ISRIB (trans-isomer), Inhibitor of “Integrated Stress Response” (ISR)
$129.00
Catalog No. M60125
A potent and selective small molecule inhibitor of PERK signaling that can potently reverse the effects of eIF2α phosphorylation, Inhibitor of “Integrated Stress Response” (ISR).
ISX9, Neurogenic ModulatorISX9, Neurogenic Modulator
ISX9, Neurogenic Modulator
$99.00
Catalog No. M60274
A neurogenic modulator.
ITD-1, TGFβ inhibitor ITD-1, TGFβ inhibitor
ITD-1, TGFβ inhibitor
$139.00
Catalog No. M60060
A highly selective TGFβ inhibitor promotes cardiomyogenesis in embryonic stem cells.
IU1, Proteasome USP14 Inhibitor IU1, Proteasome USP14 Inhibitor
IU1, Proteasome USP14 Inhibitor
$49.00
Catalog No. M60203
A cell-permeable, reversible and selective inhibitor of human proteasome USP14.
IWP-2, Porcupine (Wnt) Inhibitor IWP-2, Porcupine (Wnt) Inhibitor
IWP-2, Porcupine (Wnt) Inhibitor
$79.00
Catalog No. M60115
A potent and highly selective Wnt signaling antagonist targeting porcupine.
J147, Neuroprotective Small MoleculeJ147, Neuroprotective Small Molecule
J147, Neuroprotective Small Molecule
$89.00
Catalog No. M60012
A potent and orally active neurotrophic molecule with broadly neuroprotective efficacy in vitro and in vivo.
JIB-04 (NSC693627), Jumonji Histone Demethylase InhibitorJIB-04 (NSC693627), Jumonji Histone Demethylase Inhibitor
JIB-04 (NSC693627), Jumonji Histone Demethylase Inhibitor
$119.00
Catalog No. M60132
A potent, selective and cell permeable Jumonji histone demethylase inhibitor, not a competitive inhibitor of a-ketoglutarate.
JK184, Hedgehog Antagonist JK184, Hedgehog Antagonist
JK184, Hedgehog Antagonist
$79.00
Catalog No. M60087
A potent and cell-permeable inhibitor of hedgehog (Hh) signaling downstream of Smo.
JNJ-42041935，HIF-PHD抑制剂JNJ-42041935，HIF-PHD抑制剂
JNJ-42041935, HIF-PHD Inhibitor
$129.00
Catalog No. M60285
A potent and selective HIF-PHD inhibitor.
Kartogenin（KGN），软骨发生调节剂 Kartogenin（KGN），软骨发生调节剂
Kartogenin (KGN), Chondrogenesis Modulator
$79.00
Catalog No. M60027
Selectively promote chondrocyte differentiation of human mesenchymal stem cells.
KDM5 C70bulkKDM5 C70bulk
KDM5 C70bulk
$0.00
Catalog No. M60192-b
KDM5-C49，JARID1组蛋白脱甲基酶抑制剂 KDM5-C49，JARID1组蛋白脱甲基酶抑制剂
KDM5-C49, JARID1 Histone Demethylases Inhibitor
$139.00
Catalog No. M60191
A potent and selective inhibitor of Jumonji AT-Rich Interactive Domain 1 (JARID1) histone demethylases
KDM5-C49bulkKDM5-C49bulk
KDM5-C49bulk
$0.00
Catalog No. M60191-b
KDM5-C70，JARID1组蛋白脱甲基酶抑制剂 KDM5-C70，JARID1组蛋白脱甲基酶抑制剂
KDM5-C70, JARID1 Histone Demethylases Inhibitor
$139.00
Catalog No. M60192
An ethyl ester derivative of KDM5-C49, which is a potent and selective inhibitor of Jumonji AT-Rich Interactive Domain 1 (JARID1) histone demethylases.
KL001，Cryptochrome ActivatorKL001，Cryptochrome Activator
KL001, Cryptochrome Activator
$79.00
Catalog No. M66044
A novel small molecule specifically interacting with cryptochrome (CRY) and causing lengthening of the circadian period.
KRAS-C9，K-Ras（G12C）抑制剂 KRAS-C9，K-Ras（G12C）抑制剂
KRAS-C9, K-Ras(G12C) Inhibitor
$139.00
Catalog No. M60219
A potent and selective allosteric inhibitor of oncogenic K-Ras(G12C).
KY02111，Wnt抑制剂 KY02111，Wnt抑制剂
KY02111, Wnt Inhibitor
$109.00
Catalog No. M60073
一种有效和选择性的Wnt抑制剂促进hESC / iPSC分化成心肌细胞; 可能在β-连环蛋白破坏复合物中的GSK3β和APC的下游起作用
KYA1797K，Wnt /β-连环蛋白抑制剂KYA1797K，Wnt /β-连环蛋白抑制剂
KYA1797K，Wnt /β-连环蛋白抑制剂
$ 129.00
目录号 M60317
一种高度有效和选择性的Wnt /β-连环蛋白抑制剂直接结合轴蛋白的G蛋白信号传导结构域的调节剂。
L002（NSC764414），p300抑制剂 L002（NSC764414），p300抑制剂
L002（NSC764414），p300抑制剂
$ 99.00
目录号 M60198
一种新的选择性，细胞渗透性和可逆性p300组蛋白乙酰转移酶抑制剂。
L755,507，CRISPR编辑增强器L755,507，CRISPR编辑增强器
L755,507，CRISPR编辑增强器
$ 89.00
目录号 M60237
CRISPR编辑增强子增强人类诱导多能干细胞（iPSC）和其他细胞类型中CRISPR介导的同源性定向修复（HDR）效率。
LDE225，刺猬拮抗剂 LDE225，刺猬拮抗剂
LDE225，刺猬拮抗剂
$ 99.00
目录号 M60013
临床试验中一种有效的特异性Hedgehog通路抑制剂（Smo拮抗剂）。
LDN-193189，BMP抑制剂 LDN-193189，BMP抑制剂
LDN-193189，BMP抑制剂
$ 79.00
目录号 M60008
一种高度有效和选择性的BMP途径抑制剂（对ALK2和ALK3有选择性）; 可以在细胞和体内使用取代Noggin蛋白。
LDN-57444，泛素C-末端水解酶-L1（UCH-L1）抑制剂LDN-57444，泛素C-末端水解酶-L1（UCH-L1）抑制剂
LDN-57444，泛素C-末端水解酶-L1（UCH-L1）抑制剂
$ 69.00
目录号 M60204
泛素C端水解酶-L1（UCH-L1）的新型有效和选择性抑制剂。
LGK974，豪猪（Wnt）抑制剂 LGK974，豪猪（Wnt）抑制剂
LGK974，豪猪（Wnt）抑制剂
$ 139.00
目录号 M60106
一种高效，选择性和口服生物可利用的豪猪抑制剂（Wnt信号拮抗剂）在临床试验中。
表观遗传化合物库表观遗传化合物库
表观遗传化合物库
$ 7000.00
目录号 LI30001-2
表观遗传组合化合物库由分开的小瓶中的117个小分子组成。
LLY-507，蛋白 - 赖氨酸甲基转移酶SMYD2抑制剂LLY-507，蛋白 - 赖氨酸甲基转移酶SMYD2抑制剂
LLY-507, Protein-lysine Methyltransferase SMYD2 Inhibitor
$129.00
Catalog No. M60259
A potent, selective and cell permeable protein lysine methyltransferase SMYD2 inhibitor.
LMK235，HDAC4和HDAC5抑制剂 LMK235，HDAC4和HDAC5抑制剂
LMK235, HDAC4 and HDAC5 Inhibitor
$89.00
Catalog No. M60145
A potent and selective histone deacetylase HDAC4 and HDAC5 inhibitor.
LSD1-C76，LSD1抑制剂 LSD1-C76，LSD1抑制剂
LSD1-C76, LSD1 Inhibitor
$159.00
Catalog No. M66045
The most potent and selective Lysine Specific Demethylase-1 (LSD1) inhibitor so far.
LY2109761，TGFβ抑制剂LY2109761，TGFβ抑制剂
LY2109761, TGFβ Inhibitor
$109.00
Catalog No. M60035
A novel potent and selective TGFβ receptor type I and type II (TβRI/II) dual inhibitor with Ki of 38 nM and 300 nM respectively.
LY2157299，TGFβ抑制剂 LY2157299，TGFβ抑制剂
LY2157299, TGFβ Inhibitor
$169.00
Catalog No. M60064
A novel potent and selective TGFβ receptor type I and type II (TβRI/II) inhibitor with IC50 of 86 nM and 2 nM respectively.
LY2784544，JAK2抑制剂LY2784544，JAK2抑制剂
LY2784544, JAK2 inhibitor
$129.00
Catalog No. M60079
A highly potent and selective mutant JAK2 (V617F) inhibitor.
LY294002，PI3K / BET双重抑制剂 LY294002，PI3K / BET双重抑制剂
LY294002, PI3K/BET Dual Inhibitor
$79.00
Catalog No. M60157
A potent and selective small molecule PI3K and BET bromodomain dual inhibitor.
LY411575，γ-分泌酶抑制剂 LY411575，γ-分泌酶抑制剂
LY411575, γ-secretase Inhibitor
$119.00
Catalog No. M60078
A highly potent, selective, and orally bioavailable inhibitor of gamma secretase.
MAL-二EG-丁二酰亚胺MAL-二EG-丁二酰亚胺
MAL-di-EG-OSu
$0.00
Catalog No. L600010
Thiol reactive linker
MAL-HA-丁二酰亚胺MAL-HA-丁二酰亚胺
MAL-HA-OSu
Inquiry
Catalog No. L60005
Thiol reactive linker
MALT1-MI-2（MI-2），MALT1抑制剂 MALT1-MI-2（MI-2），MALT1抑制剂
MALT1-MI-2 (MI-2), MALT1 inhibitor
$129.00
Catalog No. M60098
A highly potent and selective small molecule directly binding to MALT1 and irreversibly suppressing its protease function.
MC1568，IIa类HDAC抑制剂MC1568，IIa类HDAC抑制剂
MC1568, Class IIa HDAC Inhibitor
$79.00
Catalog No. M60224
A potent and selective inhibitor of class IIa histone deacetylases (HDACs), more selective for HD1-A than HD1-B.
ME0328，PARP-3抑制剂ME0328，PARP-3抑制剂
ME0328, PARP-3 Inhibitor
$109.00
Catalog No. M60329
A potent, selective and cell permeable PARP-3 inhibitor.
MEK162（ARRY-162），MEK抑制剂MEK162（ARRY-162），MEK抑制剂
MEK162 (ARRY-162), MEK Inhibitor
$119.00
Catalog No. M60080
A highly potent, selective, and orally bioavailable MEK inhibitor in clinical trials.
甲氧基-XO 4，荧光淀粉样β（Aβ）探针甲氧基-XO 4，荧光淀粉样β（Aβ）探针
Methoxy-X04, Fluorescent Amyloid β (Aβ) Probe
$79.00
Catalog No. M60135
A fluorescent amyloid β (Aβ) probe for the detection and quantification of plaques, tangles and cerebrovascular amyloid with good specificity.
MHY1485，mTOR激活剂MHY1485，mTOR激活剂
MHY1485, mTOR Activator
$49.00
Catalog No. M60189
A novel potent, selective and cell-permeable mTOR activator.
MI-2，Menin-MLL抑制剂 MI-2，Menin-MLL抑制剂
MI-2, Menin-MLL Inhibitor
$119.00
Catalog No. M66046
A highly potent and selective small molecule directly binding to MALT1 and irreversibly suppressing its protease function.
MK-1775（AZD1775），WEE1抑制剂 MK-1775（AZD1775），WEE1抑制剂
MK-1775 (AZD1775), WEE1 Inhibitor
$129.00
Catalog No. M60299
A highly potent, selective and orally bioavailable Wee1 kinase inhibitor.
ML141，Cdc42 GTP酶抑制剂ML141，Cdc42 GTP酶抑制剂
ML141, Cdc42 GTPase Inhibitor
$109.00
Catalog No. M60134
A potent, selective and reversible non-competitive inhibitor of Cdc42 GTPase.
ML228，HIF通路激活剂ML228，HIF通路激活剂
ML228, HIF Pathway Activator
$129.00
Catalog No. M60130
A potent and selective hypoxia inducible factor (HIF) pathway activator.
ML239，乳腺癌干细胞抑制剂ML239，乳腺癌干细胞抑制剂
ML239, Breast Cancer Stem Cell Inhibitor
$129.00
Catalog No. M60282
A potent and selective breast cancer stem cell inhibitor.
ML323，USP1-UAF1抑制剂 ML323，USP1-UAF1抑制剂
ML323, USP1-UAF1 Inhibitor
$139.00
Catalog No. M60188
A potent, selective and reversible inhibitor of the USP1-UAF1 deubiquitinase complex.
ML324，JMJD2组蛋白脱甲基酶抑制剂 ML324，JMJD2组蛋白脱甲基酶抑制剂
ML324, JMJD2 Histone Demethylase Inhibitor
$139.00
Catalog No. M60183
A potent, selective and cell permeable inhibitor of Jumonji domain-containing protein 2 (JMJD2) histone demethylase.
MLN8237（Alisertib），Aurora A抑制剂 MLN8237（Alisertib），Aurora A抑制剂
MLN8237 (Alisertib), Aurora A inhibitor
$119.00
Catalog No. M60093
A highly potent and selective Aurora A inhibitor with >200-fold selective towards Aurora B.
MM-102，WDR5-MLL1拮抗剂MM-102，WDR5-MLL1拮抗剂
MM-102, WDR5-MLL1 Antagonist
$129.00
Catalog No. M60166
A highly potent and selective inhibitor of the MLL1/WDR5 interaction.
MRT68921，自噬激酶ULK1 / 2抑制剂 MRT68921，自噬激酶ULK1 / 2抑制剂
MRT68921, Autophagy Kinase ULK1/2 Inhibitor
$109.00
Catalog No. M60311
一种有效的，选择性和双重自噬激酶ULK1 / 2抑制剂。
MS023，PRMT抑制剂 MS023，PRMT抑制剂
MS023，PRMT抑制剂
$ 109.00
目录号 M60314
一种有效的，选择性和透过细胞的I型PRMT抑制剂。
MS049，PRMT4和PRMT6抑制剂 MS049，PRMT4和PRMT6抑制剂
MS049，PRMT4和PRMT6抑制剂
$ 89.00
目录号 M60310
一种有效的，选择性和细胞渗透性的PRMT4和PRMT6抑制剂。
MS436，BRD4抑制剂 MS436，BRD4抑制剂
MS436，BRD4抑制剂
$ 109.00
目录号 M60232
BRD4（1）和BRD4（2）是一种有效的选择性BET溴结构域抑制剂。
MSAB，β-连环蛋白抑制剂MSAB，β-连环蛋白抑制剂
MSAB，β-连环蛋白抑制剂
$ 129.00
目录号 M60316
使用基于细胞的化学筛选鉴定了一种有效和选择性的Wnt /β-连环蛋白抑制剂。
N106，SERCA2a SUMOylation活化剂N106，SERCA2a SUMOylation活化剂
N106，SERCA2a SUMOylation活化剂
$ 129.00
目录号 M60271
一种有效的SERCA2a SUMOylation活化剂，可增加SERCA2a的SUMO化。
N3三EG-OSu的N3三EG-OSu的
N3三EG-OSu的
查询
目录号 L60004
点击化学链接器
NAB2，Rsp5 / Nedd4通路激活剂，拯救α-突触核蛋白毒性NAB2，Rsp5 / Nedd4通路激活剂，拯救α-突触核蛋白毒性
NAB2，Rsp5 / Nedd4通路激活剂，拯救α-突触核蛋白毒性
$ 129.00
目录号 M60153
一种新型且高效的小分子Rsp5 / Nedd4通路激活剂，被证明能够强有力地选择性地保护不同类型的细胞免受α-突触核蛋白毒性。
Napabucasin（BBI608），STAT3抑制剂Napabucasin（BBI608），STAT3抑制剂
Napabucasin（BBI608），STAT3抑制剂
$ 89.00
目录号 M60303
一种有效和选择性的STAT3抑制剂。
神经LSB神经LSB
神经LSB
$ 79.00
目录号 S10001
LDN193189（BMP抑制剂）和SB431542（TGFβ抑制剂）的组合可以在5天内快速且有效地诱导人ESC和iPSC的神经分化。
神经细胞 - LSB3i神经细胞 - LSB3i
神经细胞 - LSB3i
$ 329.00
目录号 S10002
Combination of LSB and three other inhibitors/3i (i.e., CHIR99021/GSK3 inhibitor, SU5402/FGF-VEGF-PDGF inhibitor, DAPT/Notch inhibitor) can induce very rapid and efficient neuronal differentiation of human ESC and iPSC into nociceptors.
NI-57，BRPF溴代域抑制剂NI-57，BRPF溴代域抑制剂
NI-57, BRPF Bromodomain Inhibitor
$109.00
Catalog No. M60279
A potent and selective inhibitor of the bromodomain of the BRPFs.
NLG919 (RG6078), IDO InhibitorNLG919 (RG6078), IDO Inhibitor
NLG919 (RG6078), IDO Inhibitor
$129.00
Catalog No. M60258
A potent, selective and orally bioavailable IDO (indoleamine-(2,3)-dioxygenase) pathway inhibitor.
NMS-859, ATPase VCP/p97 InhibitorNMS-859, ATPase VCP/p97 Inhibitor
NMS-859, ATPase VCP/p97 Inhibitor
$139.00
Catalog No. M60148
A potent and specific small molecule covalent inhibitor of the ATPase VCP/p97.
NMS-873, ATPase VCP/p97 Inhibitor NMS-873, ATPase VCP/p97 Inhibitor
NMS-873, ATPase VCP/p97 Inhibitor
$139.00
Catalog No. M60165
A potent and specific small molecule allosteric inhibitor of the ATPase VCP/p97.
NMS-873/BulkNMS-873/Bulk
NMS-873/Bulk
$0.00
Catalog No. M60165-b
Nocodazole, Microtubule Inhibitor / CRISPR Editing EnhancerNocodazole, Microtubule Inhibitor / CRISPR Editing Enhancer
Nocodazole, Microtubule Inhibitor / CRISPR Editing Enhancer
$79.00
Catalog No. M60331
A potent microtubule inhibitor to inhibit mitosis and CRISPR editing enhancer.
NSC319726, Mutant p53 Activator NSC319726, Mutant p53 Activator
NSC319726, Mutant p53 Activator
$89.00
Catalog No. M66047
A potent and selective activator of the most common p53R175 mutant, restoring the mutant p53 to its WT structure and function.
NSC636819, KDM4A/KDM4B InhibitorNSC636819, KDM4A/KDM4B Inhibitor
NSC636819, KDM4A/KDM4B Inhibitor
$109.00
Catalog No. M60290
A cell permeable and selective novel active-site KDM4A/KDM4B inhibitor.
NSC697923, Ub-conjugating Enzyme (E2) InhibitorNSC697923, Ub-conjugating Enzyme (E2) Inhibitor
NSC697923, Ub-conjugating Enzyme (E2) Inhibitor
$69.00
Catalog No. M60202
A cell permeable, potent and selective inhibitor of the Ub-conjugating enzyme (E2) complex Ubc13-Uev1A.
NU9056--- KAT5 (Tip60) Histone Acetyltransferase InhibitorNU9056--- KAT5 (Tip60) Histone Acetyltransferase Inhibitor
NU9056--- KAT5 (Tip60) Histone Acetyltransferase Inhibitor
$69.00
Catalog No. M60147
A potent and selective KAT5 (Tip60) histone acetyltransferase inhibitor.
NVP-BGT226, PI3K/mTOR Dual InhibitorNVP-BGT226, PI3K/mTOR Dual Inhibitor
NVP-BGT226, PI3K/mTOR Dual Inhibitor
$89.00
Catalog No. M66050
A PI3K/mTOR dual inhibitor in clinical trials for advanced solid tumors.
NVP-BKM120, PI3K Inhibitor BKM120NVP-BKM120, PI3K Inhibitor BKM120
NVP-BKM120, PI3K Inhibitor BKM120
$89.00
Catalog No. M66051
A selective PI3K Inhibitor in clinical trials for advanced solid tumors.
NVP-TNKS656, Wnt / Tankyrase Inhibitor NVP-TNKS656, Wnt / Tankyrase Inhibitor
NVP-TNKS656, Wnt / Tankyrase Inhibitor
$109.00
Catalog No. M60328
A highly potent, selective and oral bioavailable tankyrase inhibitor for TNKS2.
NVS-SM1, SMN2 Splicing ModulatorNVS-SM1, SMN2 Splicing Modulator
NVS-SM1, SMN2 Splicing Modulator
$129.00
Catalog No. M60277
A highly potent, selective and orally active small molecule SMN2 splicing modulator enhancing SMN exon 7 inclusion.
NVS-SM1BulkNVS-SM1Bulk
NVS-SM1Bulk
$0.00
Catalog No. M60277-b
OAC1, Oct4 ActivatorOAC1, Oct4 Activator
OAC1, Oct4 Activator
$109.00
Catalog No. M60086
A potent Oct4 activator significantly enhancing iPSC reprogramming efficiency and accelerating the reprogramming process.
OF-1, BRPF Bromodomain Inhibitor OF-1, BRPF Bromodomain Inhibitor
OF-1, BRPF Bromodomain Inhibitor
$129.00
Catalog No. M60222
A potent and selective BRPF (BRomodomain and PHD Finger containing) inhibitor.
OG-L002, LSD1 InhibitorOG-L002, LSD1 Inhibitor
OG-L002, LSD1 Inhibitor
$89.00
Catalog No. M60161
A highly potent and specific inhibitor of Lysine Specific Demethylase-1 (LSD1).
OICR9429, WDR5 AntagonistOICR9429, WDR5 Antagonist
OICR9429, WDR5 Antagonist
$129.00
Catalog No. M60255
A potent and selective WD repeat-containing protein 5 (WDR5) antagonist.
ONX-0914, Immunoproteasome InhibitorONX-0914, Immunoproteasome Inhibitor
ONX-0914, Immunoproteasome Inhibitor
$139.00
Catalog No. M60112
A potent and selective immunoproteasome inhibitor.
Optovin, TRPA1 ActivatorOptovin, TRPA1 Activator
Optovin, TRPA1 Activator
$129.00
Catalog No. M60103
A potent and selective small molecule activator of human TRPA1.
ORY-1001 (RG-6016), LSD1 InhibitorORY-1001 (RG-6016), LSD1 Inhibitor
ORY-1001 (RG-6016), LSD1 Inhibitor
$129.00
Catalog No. M60295
A highly potent and selective inhibitor of Lysine Specific Demethylase 1 (LSD1) in phase I/II.
OSI-027, mTOR InhibitorOSI-027, mTOR Inhibitor
OSI-027, mTOR Inhibitor
$109.00
Catalog No. M60113
OSI-027 is a selective and potent dual inhibitor of mTORC1 and mTORC2
OTX015, BET Inhibitor OTX015, BET Inhibitor
OTX015, BET Inhibitor
$89.00
Catalog No. M60193
OTX015 is a novel, highly potent, selective and cell permeable inhibitor of the bromodomain and extra terminal (BET) family proteins BRD2, BRD3 and BRD4 with IC50 of 10-19 nM.
P22077, USP7 inhibitorP22077, USP7 inhibitor
P22077, USP7 inhibitor
$99.00
Catalog No. M60019
A potent and selective USP7 inhibitor.
P5091, Ubiquitin-specific Protease 7 (USP7) InhibitorP5091, Ubiquitin-specific Protease 7 (USP7) Inhibitor
P5091, Ubiquitin-specific Protease 7 (USP7) Inhibitor
$79.00
Catalog No. M60205
P5091 (P005091) is a novel potent and selective inhibitor of ubiquitin-specific protease 7 (USP7)
P7C3, Neuroprotective Small MoleculeP7C3, Neuroprotective Small Molecule
P7C3, Neuroprotective Small Molecule
$119.00
Catalog No. M60017
A neuroprotective small molecule with favorable in vivo PK; protects newborn neurons from apoptosis.
PBIT，JARID1组蛋白脱甲基酶抑制剂PBIT，JARID1组蛋白脱甲基酶抑制剂
PBIT, JARID1 Histone Demethylases Inhibitor
$129.00
Catalog No. M60170
PBIT is a potent, specific, reversible and cell-permeable inhibitor of Jumonji AT-Rich Interactive Domain 1 (JARID1) histone demethylases.
PCI-34051，HDAC8抑制剂PCI-34051，HDAC8抑制剂
PCI-34051, HDAC8 Inhibitor
$79.00
Catalog No. M60178
PCI-34051 is a potent and selective inhibitor of histone deacetylase 8 (HDAC8).
PD-1 / PD-L1抑制剂C1PD-1 / PD-L1抑制剂C1
PD-1/PD-L1 Inhibitor C1
$109.00
Catalog No. M60312
PD-1 / PD-L1蛋白/蛋白质相互作用的有效和选择性小分子抑制剂。
PD0325901，MEK抑制剂PD0325901，MEK抑制剂
PD0325901，MEK抑制剂
$ 69.00
目录号 M60018
一种有效和选择性的MEK抑制剂。
PF-04979064，PI3K / mTOR双重抑制剂PF-04979064，PI3K / mTOR双重抑制剂
PF-04979064，PI3K / mTOR双重抑制剂
$ 149.00
目录号 M60114
PF-04979064是一种高效且口服生物可利用的PI3K / mTOR双重抑制剂，通过基于结构的**设计开发。
PF-CBP1，CBP / p300溴代域抑制剂 PF-CBP1，CBP / p300溴代域抑制剂
PF-CBP1，CBP / p300溴代域抑制剂
$ 129.00
目录号 M60313
一种有效和选择性的CBP / p300溴结构域抑制剂。
PFI-1，BET抑制剂PFI-1，BET抑制剂
PFI-1，BET抑制剂
$ 129.00
目录号 M60120
PFI-1是溴结构域和额外终端（BET）家族蛋白BRD2和BRD4的新型有效，选择性和细胞渗透性抑制剂。
PFI-2，SETD7组蛋白赖氨酸甲基转移酶抑制剂 PFI-2，SETD7组蛋白赖氨酸甲基转移酶抑制剂
PFI-2，SETD7组蛋白赖氨酸甲基转移酶抑制剂
$ 139.00
目录号 M60182
PFI-2是一种新型强效和选择性SETD7组蛋白赖氨酸甲基转移酶抑制剂。
PFI-3，SMARCA Bromodomains抑制剂PFI-3，SMARCA Bromodomains抑制剂
PFI-3，SMARCA Bromodomains抑制剂
$ 139.00
目录号 M60175
PFI-3是SMARCA4和PB1（5）溴结构域的新型有效，选择性和细胞渗透性抑制剂。
PFI-4，BRPF1溴结构域抑制剂PFI-4，BRPF1溴结构域抑制剂
PFI-4，BRPF1溴结构域抑制剂
$ 129.00
目录号 M60264
一种有效的，选择性和细胞渗透性的BRPF1溴结构域抑制剂。
磷酸-HDAC4（Ser632）抗体磷酸-HDAC4（Ser632）抗体
磷酸-HDAC4（Ser632）抗体
$ 0.00包装
目录号 A90009-5
一个
磷酸-HDAC4（Ser632）抗体磷酸-HDAC4（Ser632）抗体
磷酸-HDAC4（Ser632）抗体
$ 0.00包装
目录号 A90009
磷酸-HDAC4（Ser632）抗体。组蛋白去乙酰化酶4（HDAC4）是一种组蛋白脱乙酰酶，其在连接到启动子时抑制转录。
PluriSIn＃1，多能细胞特异性抑制剂 PluriSIn＃1，多能细胞特异性抑制剂
PluriSIn＃1，多能细胞特异性抑制剂
$ 109.00
目录号 M60085
A potent small molecule to selectively eliminate human pluripotent stem cells/hPSCs while sparing a large array of tissue-specific stem/progenitor and differentiated cells.
pNSC-CSBpNSC-CSB
pNSC-CSB
$69.00
Catalog No. S10003
Combination of CHIR99021 (GSK3 inhibitor) and SB431542 (TGFβ inhibitor) with human LIF can efficiently induce and long-term homogenously expand primitive neural stem cells from human ESC and iPSC.
PP242，mTORC1 / mTORC2抑制剂PP242，mTORC1 / mTORC2抑制剂
PP242, mTORC1/mTORC2 inhibitor
$69.00
Catalog No. M60094
A highly potent, selective and ATP-competitive mTORC1/mTORC2 inhibitor.
PR-619，去泛素化酶（DUB）抑制剂 PR-619，去泛素化酶（DUB）抑制剂
PR-619, Deubiquitinylating Enzyme (DUB) Inhibitor
$59.00
Catalog No. M60199
PR-619 is a cell-permeable, non-selective, reversible broad-range inhibitor of the deubiquitinylating enzymes (DUBs).
PRMT1-2e，蛋白精氨酸甲基转移酶1（PRMT1）抑制剂 PRMT1-2e，蛋白精氨酸甲基转移酶1（PRMT1）抑制剂
PRMT1-2e, Protein Arginine Methyltransferase 1 (PRMT1) Inhibitor
$69.00
Catalog No. M60181
PRMT1-2e is a potent, specific and cell permeable inhibitor of protein arginine methyltransferase 1 (PRMT1).
PRT4165，E3泛素连接酶Bmi1 / Ring1A抑制剂PRT4165，E3泛素连接酶Bmi1 / Ring1A抑制剂
PRT4165, E3 Ubiquitin-ligase Bmi1/Ring1A Inhibitor
$39.00
Catalog No. M60245
A potent and selective E3 Ubiquitin-ligase Bmi1/Ring1A Inhibitor.
PS48 --- PDK1 ActivatorPS48 --- PDK1 Activator
PS48---PDK1 Activator
$79.00
Catalog No. M60026
An allosteric small molecule activator of PDK1.
PTC-209，BMI-1抑制剂PTC-209，BMI-1抑制剂
PTC-209, BMI-1 Inhibitor
$129.00
Catalog No. M60159
PTC-209 is a novel potent and selective BMI-1 inhibitor, targeting the BMI-1 self-renewal machinery.
PTC-209BulkPTC-209Bulk
PTC-209Bulk
$0.00
Catalog No. M60159-b
Purmorphamine，刺猬激动剂 Purmorphamine，刺猬激动剂
Purmorphamine, Hedgehog Agonist
$99.00
Catalog No. M66055
A selective hedgehog pathway agonist (Smo agonist).
PX-478，缺氧诱导因子-1α（HIF-1α）抑制剂 PX-478，缺氧诱导因子-1α（HIF-1α）抑制剂
PX-478, Hypoxia-inducible Factor-1α (HIF-1α) Inhibitor
$129.00
Catalog No. M60227
A highly potent and selective Hypoxia-inducible Factor-1α (HIF-1α) inhibitor.
PY-DS-但是，丁二酰亚胺PY-DS-但是，丁二酰亚胺
Py-ds-But-OSu
Inquiry
Catalog No. L60003
Disulfide prodrug linker
PYR-41 ---泛素激活酶E1抑制剂 PYR-41 ---泛素激活酶E1抑制剂
PYR-41---Ubiquitin-activating Enzyme E1 Inhibitor
$59.00
Catalog No. M60201
PYR-41 is a specific and cell permeable inhibitor of ubiquitin-activating enzyme E1
Pyrintegrin---Cell Survival EnhancerPyrintegrin---Cell Survival Enhancer
Pyrintegrin---Cell Survival Enhancer
$109.00
Catalog No. M60028
A potent small molecule promoting hESC survival
PYZD-4409, Ubiquitin-activating Enzyme (E1) Inhibitor PYZD-4409, Ubiquitin-activating Enzyme (E1) Inhibitor
PYZD-4409, Ubiquitin-activating Enzyme (E1) Inhibitor
$139.00
Catalog No. M60213
A novel potent, selective and cell permeable inhibitor of ubiquitin-activating enzyme (E1).
RA190, Ubiquitin Receptor RPN13/ADRM1 InhibitorRA190, Ubiquitin Receptor RPN13/ADRM1 Inhibitor
RA190, Ubiquitin Receptor RPN13/ADRM1 Inhibitor
$139.00
Catalog No. M60163
A novel potent and selective inhibitor of proteasome Ubiquitin receptor RPN13/ADRM1.
RA190bulkRA190bulk
RA190bulk
$0.00
Catalog No. M60163-b
Rapamycin, mTOR inhibitor Rapamycin, mTOR inhibitor
Rapamycin, mTOR inhibitor
$89.00
Catalog No. M60029
A potent and selective mTOR inhibitor, directly binding to the mTOR Complex 1 (mTORC1).
Recombinant Human Activin ARecombinant Human Activin A
Recombinant Human Activin A
$3900.00
Catalog No. G2001601-1MG
n/a
Recombinant Human Basic Fibroblast Growth FactorRecombinant Human Basic Fibroblast Growth Factor
Recombinant Human Basic Fibroblast Growth Factor
$995.00
Catalog No. G2001602-1MG
n/a
Recombinant Human Epidermal Growth FactorRecombinant Human Epidermal Growth Factor
Recombinant Human Epidermal Growth Factor
$140.00
Catalog No. G2001603-1MG
n/a
Recombinant Human Insulin-like Growth Factor-1Recombinant Human Insulin-like Growth Factor-1
Recombinant Human Insulin-like Growth Factor-1
$235.00
Catalog No. G2001604-1MG
n/a
Recombinant Human Platelet-Derived Growth Factor-BBRecombinant Human Platelet-Derived Growth Factor-BB
Recombinant Human Platelet-Derived Growth Factor-BB
$3200.00
Catalog No. G2001605-1MG
n/a
Recombinant Human Transforming Growth Factor,Beta 1Recombinant Human Transforming Growth Factor,Beta 1
Recombinant Human Transforming Growth Factor,Beta 1
$5050.00
Catalog No. G2001606-1MG
n/a
Recombinant Mouse Basic Fibroblast Growth FactorRecombinant Mouse Basic Fibroblast Growth Factor
Recombinant Mouse Basic Fibroblast Growth Factor
$880.00
Catalog No. G2001652-1MG
n/a
Recombinant Mouse Epidermal Growth FactorRecombinant Mouse Epidermal Growth Factor
Recombinant Mouse Epidermal Growth Factor
$220.00
Catalog No. G2001653-1MG
n/a
Recombinant Mouse Leukemia Inhibitory FactorRecombinant Mouse Leukemia Inhibitory Factor
Recombinant Mouse Leukemia Inhibitory Factor
$2640.00
Catalog No. G2001651-1MG
n/a
Remodelin, Acetyl-transferase NAT10 InhibitorRemodelin, Acetyl-transferase NAT10 Inhibitor
Remodelin, Acetyl-transferase NAT10 Inhibitor
$139.00
Catalog No. M60187
Remodelin is a novel potent and selective inhibitor of the acetyl-transferase protein NAT10.
RepSox---TGF-β Type I Receptor ALK5 Inhibitor RepSox---TGF-β Type I Receptor ALK5 Inhibitor
RepSox---TGF-β Type I Receptor ALK5 Inhibitor
$79.00
Catalog No. M60151
RepSox (E-616452 or SJN 2511) is a highly potent, selective inhibitor of the TGF-β type I receptor ALK5.
RG108---DNA Methyltransferase InhibitorRG108---DNA Methyltransferase Inhibitor
RG108---DNA Methyltransferase Inhibitor
$65.00
Catalog No. M60176
RG108 is a potent, selective and cell permeable inhibitor of DNA methyltransferase.
RG2833 (RGFP109), Brain-penetrant HDAC InhibitorRG2833 (RGFP109), Brain-penetrant HDAC Inhibitor
RG2833 (RGFP109), Brain-penetrant HDAC Inhibitor
$69.00
Catalog No. M60225
A potent and selective brain-penetrant HDAC inhibitor HDAC1 and HDAC3.
RGFP966, HDAC3 Inhibitor RGFP966, HDAC3 Inhibitor
RGFP966, HDAC3 Inhibitor
$89.00
Catalog No. M60156
RGFP966 is a potent and selective HDAC3 inhibitor.
RN-1, LSD1 Inhibitor RN-1, LSD1 Inhibitor
RN-1, LSD1 Inhibitor
$109.00
Catalog No. M60169
RN-1 is a potent, specific and brain-penetrant Lysine Specific Demethylase-1 (LSD1) inhibitor.
RO4929097, γ-Secretase InhibitorRO4929097, γ-Secretase Inhibitor
RO4929097, γ-Secretase Inhibitor
$109.00
Catalog No. M60007
A potent and selective γ-secretase inhibitor; inhibits Notch signaling in stem cells and tumor cells.
RS-1, CRISPR Editing Enhancer RS-1, CRISPR Editing Enhancer
RS-1, CRISPR Editing Enhancer
$89.00
Catalog No. M60300
Previously characterized as a RAD51-Stimulatory compound and now found to be an HDR enhancer to enhance CRISPR/Cas9- and TALEN-mediated knock-in efficiency
RU-SKI 43，Hhat抑制剂RU-SKI 43，Hhat抑制剂
RU-SKI 43, Hhat Inhibitor
$139.00
Catalog No. M60100
The first potent and specific small molecule inhibitor of Hedgehog acyltransferase (Hhat).
RVX-208，BET溴代域抑制剂RVX-208，BET溴代域抑制剂
RVX-208, BET Bromodomain Inhibitor
$59.00
Catalog No. M60177
RVX-208 is a potent and selective BET bromodomain inhibitor for the second bromodomain (BD2), ~170-fold selectivity over BD1.
龙血素，赖氨酸甲基转移酶SETD8抑制剂龙血素，赖氨酸甲基转移酶SETD8抑制剂
Ryuvidine, Lysine Methyltransferase SETD8 Inhibitor
$129.00
Catalog No. M60252
A potent, selective and cell permeable lysine methyltransferase SETD8 inhibitor.
SAG，刺猬激动剂SAG，刺猬激动剂
SAG, Hedgehog Agonist
$129.00
Catalog No. M60081
A potent, selective, and cell-permeable small-molecule agonist of the Hedgehog pathway.
SB431542，TGF-β抑制剂SB431542，TGF-β抑制剂
SB431542，TGF-β抑制剂
$ 300.00
目录号 M60015
一种有效的选择性TGF-β途径抑制剂（对ALK4，ALK5和ALK7具有选择性）。
SBI-0206965，自噬激酶ULK1抑制剂SBI-0206965，自噬激酶ULK1抑制剂
SBI-0206965，自噬激酶ULK1抑制剂
$ 129.00
目录号 M60268
一种有效的，选择性和细胞渗透性自噬激酶ULK1抑制剂。
SCH51344，MTH1抑制剂 SCH51344，MTH1抑制剂
SCH51344，MTH1抑制剂
$ 139.00
目录号 M60212
一种新型有效的，选择性和细胞渗透性的MTH1抑制剂。
SCR7，NHEJ抑制剂SCR7，NHEJ抑制剂
SCR7，NHEJ抑制剂
$ 129.00
目录号 M60082
一种有效的选择性非同源末端连接抑制剂（NHEJ）。
SD70，组蛋白脱甲基酶JMJD2抑制剂 SD70，组蛋白脱甲基酶JMJD2抑制剂
SD70，组蛋白脱甲基酶JMJD2抑制剂
$ 139.00
目录号 M60194
一种有效的，选择性和细胞渗透性的组蛋白去甲基化酶JMJD2（KDM4C）抑制剂。
Sephin1，PPP1R15A蛋白磷酸酶抑制剂Sephin1，PPP1R15A蛋白磷酸酶抑制剂
Sephin1，PPP1R15A蛋白磷酸酶抑制剂
$ 129.00
目录号 M60280
蛋白磷酸酶1的调节亚基PPP1R15A的有效的，选择性的和生物可利用的抑制剂。
SGC-CBP30，p300 / CBP溴代域抑制剂 SGC-CBP30，p300 / CBP溴代域抑制剂
SGC-CBP30，p300 / CBP溴代域抑制剂
$ 139.00
目录号 M60138
SGC-CBP30是一种高度有效和选择性的p300 / CBP bromodomain抑制剂
SGC0946，DOT1L抑制剂 SGC0946，DOT1L抑制剂
SGC0946，DOT1L抑制剂
$ 139.00
目录号 M60101
DOT1L甲基转移酶的高度有效和选择性抑制剂。
SGC707，变构PRMT3抑制剂SGC707，变构PRMT3抑制剂
SGC707，变构PRMT3抑制剂
$ 129.00
目录号 M60243
一种有效的，选择性和细胞渗透性变构蛋白精氨酸甲基转移酶3（PRMT3）抑制剂。
SGI-1027，DNMT抑制剂SGI-1027，DNMT抑制剂
SGI-1027，DNMT抑制剂
$ 89.00
目录号 M60155
一种有效的选择性DNA甲基转移酶抑制剂（DNMT）。
SHP099，SHP2磷酸酶抑制剂SHP099，SHP2磷酸酶抑制剂
SHP099，SHP2磷酸酶抑制剂
$ 139.00
目录号 M60319
A highly potent, selective and orally bioavailable small-molecule SHP2 inhibitor.
SirReal2，Sirt2抑制剂SirReal2，Sirt2抑制剂
SirReal2, Sirt2 Inhibitor
$119.00
Catalog No. M60289
A potent and selective Sirt2 inhibitor.
SIRT1多克隆抗体SIRT1多克隆抗体
SIRT1 Polyclonal Antibody
$0.00
Catalog No. A90007
SIRT1 Polyclonal Antibody: SIRT1 is a nuclear protein that regulates epigenetic gene silencing and suppresses recombination of rDNA
SKP2-C25，Skp2抑制剂SKP2-C25，Skp2抑制剂
SKP2-C25, Skp2 Inhibitor
$139.00
Catalog No. M60136
A potent, selective and cell permeable Skp2 inhibitor, selectively inhibits Skp2 E3 ligase activity, but not activity of other SCF complexes.
SKPin C1，Skp2抑制剂 SKPin C1，Skp2抑制剂
SKPin C1, Skp2 Inhibitor
$109.00
Catalog No. M60137
A potent and selective inhibitor of Skp2-mediated p27 degradation.
SMER3，SCF家族E3泛素连接酶抑制剂 SMER3，SCF家族E3泛素连接酶抑制剂
SMER3, SCF family E3 Ubiquitin Ligase Inhibitor
$129.00
Catalog No. M60250
A potent and selective a yeast SCF family E3 ubiquitin ligase inhibitor, also a small-molecule enhancers of rapamycin.
Spautin-1，自噬抑制剂Spautin-1，自噬抑制剂
Spautin-1, Autophagy Inhibitor
$69.00
Catalog No. M60003
A potent autophagy inhibitor, selectively promotes the degradation of Vps34 complexes.
SR10067，REV-ERB激动剂SR10067，REV-ERB激动剂
SR10067, REV-ERB Agonist
$129.00
Catalog No. M60240
A potent and specific synthetic REV-ERB agonist.
SR1664，PPAR-γ调制器SR1664，PPAR-γ调制器
SR1664,PPAR-γ Modulator
$109.00
Catalog No. M66048
An unique PPARγ modulator that has potent anti-diabetic activity through blocking the Cdk5-mediated phosphorylation of PPARγ, but completely lacks classical transcriptional agonism that accounts for other PPARγ agonists’ side effects.
SR9009，REV-ERB激动剂SR9009，REV-ERB激动剂
SR9009, REV-ERB Agonist
$109.00
Catalog No. M60236
A potent and specific synthetic REV-ERB agonist.
SR9011SR9011
SR9011
$1250.00
Catalog No. M66049-b
SR9011，REV-ERB激动剂SR9011，REV-ERB激动剂
SR9011, REV-ERB Agonist
$109.00
Catalog No. M66049
A potent synthetic REV-ERB agonist with in vivo activity; can regulate circadian behavior and metabolism.
SR9011-CSR9011-C
SR9011-c
$1250.00
Catalog No. SR9011-c
SR9243，LXR反激动剂SR9243，LXR反激动剂
SR9243, LXR Inverse Agonist
$129.00
Catalog No. M60270
A highly potent and selective small molecule LXR inverse agonist that induces LXR-corepressor interaction.
StemRegenin1（SR1）--- HSC扩增分子StemRegenin1（SR1）--- HSC扩增分子
StemRegenin1 (SR1)---HSC Expansion Molecule
$99.00
Catalog No. M60001
A potent and selective aryl hydrocarbon receptor antagonist; can promote robust expansion of human CD34+ hematopoietic stem and progenitor cells.
SU5402 --- FGFR抑制剂 SU5402 --- FGFR抑制剂
SU5402---FGFR inhibitor
$89.00
Catalog No. M60025
A potent and selective inhibitor of FGFR, VEGFR, and PDGFR.
SW033291,15-PGDH抑制剂SW033291,15-PGDH抑制剂
SW033291, 15-PGDH Inhibitor
$99.00
Catalog No. M60298
一种高度有效的选择性15-PGDH抑制剂，可增加骨髓和其他组织中前列腺素PGE2的水平。
TAK-243（MLN7243），泛素活化酶（UAE）抑制剂 TAK-243（MLN7243），泛素活化酶（UAE）抑制剂
TAK-243（MLN7243），泛素活化酶（UAE）抑制剂
$ 129.00
目录号 M60332
泛素活化酶（UAE）的一种有效的，选择性和细胞渗透性的小分子抑制剂。
TAK-875（Fasiglifam），GPR40激动剂TAK-875（Fasiglifam），GPR40激动剂
TAK-875（Fasiglifam），GPR40激动剂
$ 139.00
目录号 M60220
一种有效的，选择性和口服生物可利用的部分GPR40激动剂。
TAME，泛素连接酶APC / C抑制剂TAME，泛素连接酶APC / C抑制剂
TAME，泛素连接酶APC / C抑制剂
$ 29.00
目录号 M60246
泛素连接酶后期促进复合体/细胞体（APC / C）的竞争性抑制剂。
Tasquinimod，变构HDAC4抑制剂Tasquinimod，变构HDAC4抑制剂
Tasquinimod，变构HDAC4抑制剂
$ 129.00
目录号 M60235
一种有效的选择性变构HDAC4抑制剂。
TCID，泛素C-末端水解酶-L3（UCH-L3）抑制剂 TCID，泛素C-末端水解酶-L3（UCH-L3）抑制剂
TCID，泛素C-末端水解酶-L3（UCH-L3）抑制剂
$ 99.00
目录号 M60197
泛素C-端水解酶-L3（UCH-L3）的新型有效和选择性抑制剂
TEPP-46（ML265），丙酮酸激酶M2（PKM2）激活剂TEPP-46（ML265），丙酮酸激酶M2（PKM2）激活剂
TEPP-46（ML265），丙酮酸激酶M2（PKM2）激活剂
$ 129.00
目录号 M60304
一种有效的选择性丙酮酸激酶M2（PKM2）激活剂。
TG101348（SAR302503），JAK2和BRD4双重抑制剂 TG101348（SAR302503），JAK2和BRD4双重抑制剂
TG101348（SAR302503），JAK2和BRD4双重抑制剂
$ 109.00
目录号 M60172
在临床试验中，TG101348是JAK2和BRD4的一种有效的，特异性的和口服生物可利用的抑制剂。
TH-302，缺氧激活的前药TH-302，缺氧激活的前药
TH-302，缺氧激活的前药
$ 179.00
目录号 M60089
一种高度有效且选择性低氧激活的前药靶向实体瘤的缺氧区域。
TH588，MTH1抑制剂TH588，MTH1抑制剂
TH588，MTH1抑制剂
$ 139.00
目录号 M60211
一种新型有效的，选择性和细胞渗透性的MTH1抑制剂。
Thiazovivin，岩石抑制剂 Thiazovivin，岩石抑制剂
Thiazovivin，岩石抑制剂
$ 79.00
目录号 M60009
A more potent and selective Rock inhibitor; can enhance hESC and hiPSC survival from single cell dissociation.
THZ1，共价CDK7抑制剂THZ1，共价CDK7抑制剂
THZ1, Covalent CDK7 Inhibitor
$159.00
Catalog No. M60214
A novel potent, selective and cell permeable irreversible CDK7 inhibitor.
TMP269，IIa类HDAC抑制剂TMP269，IIa类HDAC抑制剂
TMP269, Class IIa HDAC Inhibitor
$129.00
Catalog No. M60119
A highly potent, selective and cell-permeable class IIa HDAC inhibitor.
TMPA --- AMPK活化剂TMPA --- AMPK活化剂
TMPA---AMPK Activator
$119.00
Catalog No. M60072
TMPA is a novel small molecule that binds to orphan Nuclear Receptor Nur77 and activates AMPK.
TRIM24-C34，BRPF1B / TRIM24双重抑制剂TRIM24-C34，BRPF1B / TRIM24双重抑制剂
TRIM24-C34, BRPF1B/TRIM24 Dual Inhibitor
$99.00
Catalog No. M60265
A potent, selective and cell permeable BRPF1B and TRIM24 dual inhibitor.
TRIM24-C34bulkTRIM24-C34bulk
TRIM24-C34bulk
$169.00 $199.00
Catalog No. M60265-b
TRIM24-C34bulkTRIM24-C34bulk
TRIM24-C34bulk
$0.00
Catalog No. M60265-b
TZ9，Rad6泛素抑制剂 TZ9，Rad6泛素抑制剂
TZ9, Rad6 Ubiquitin Inhibitor
$109.00
目录号 M60286
人类E2泛素缀合酶Rad6B的选择性和细胞渗透性抑制剂。
UF010，HDAC抑制剂UF010，HDAC抑制剂
UF010，HDAC抑制剂
$ 89.00
目录号 M60278
UF010是一种有效的选择性I类HADC抑制剂。
UM171，人类HSC自我更新激动剂UM171，人类HSC自我更新激动剂
UM171，人类HSC自我更新激动剂
$ 159.00
目录号 M60223
刺激人体脐带血细胞体外扩增的有效小分子能够在**功能低下的小鼠中重建人造血系统至少6个月。
UNC0379，赖氨酸甲基转移酶SETD8抑制剂 UNC0379，赖氨酸甲基转移酶SETD8抑制剂
UNC0379，赖氨酸甲基转移酶SETD8抑制剂
$ 129.00
目录号 M60207
赖氨酸甲基转移酶SETD8的新型选择性，底物竞争性抑制剂
UNC0638，G9a HMTase抑制剂 UNC0638，G9a HMTase抑制剂
UNC0638，G9a HMTase抑制剂
$ 89.00
目录号 M66056
G9a（EHMT2）和GLP（EHMT1）组蛋白甲基转移酶的有效，选择性和细胞渗透性抑制剂。
UNC0642，G9a / GLP HMTase抑制剂 UNC0642，G9a / GLP HMTase抑制剂
UNC0642，G9a / GLP HMTase抑制剂
$ 129.00
目录号 M60185
同源蛋白赖氨酸甲基转移酶G9a和GLP的一种新型高效，选择性和细胞渗透性抑制剂，具有改善的PK特性。
UNC0646，G9a / GLP HMTase抑制剂 UNC0646，G9a / GLP HMTase抑制剂
UNC0646，G9a / GLP HMTase抑制剂
$ 89.00
目录号 M60184
一种新的有效的，选择性和细胞渗透性同源蛋白赖氨酸甲基转移酶G9a和GLP抑制剂。
UNC1215，L3MBTL3域抑制剂UNC1215，L3MBTL3域抑制剂
UNC1215，L3MBTL3域抑制剂
$ 119.00
目录号 M60084
用于L3MBTL3的甲基赖氨酸（Kme）阅读功能的高度有效和选择性的小分子抑制剂。
UNC2170，甲基赖氨酸结合蛋白53BP1抑制剂UNC2170，甲基赖氨酸结合蛋白53BP1抑制剂
UNC2170，甲基赖氨酸结合蛋白53BP1抑制剂
$ 99.00
目录号 M60260
选择性和细胞渗透性甲基赖氨酸结合蛋白53BP1拮抗剂。
UNC2327，变构PRMT3抑制剂 UNC2327，变构PRMT3抑制剂
UNC2327，变构PRMT3抑制剂
$ 129.00
目录号 M60253
一种有效的选择性变构蛋白精氨酸甲基转移酶3（PRMT3）抑制剂。
UNC669，L3MBTL1域抑制剂 UNC669，L3MBTL1域抑制剂
UNC669，L3MBTL1域抑制剂
$ 89.00
目录号 M60083
用于L3MBTL1的甲基赖氨酸（Kme）阅读功能的有效和选择性小分子抑制剂
维替泊芬（Visudyne），YAP抑制剂维替泊芬（Visudyne），YAP抑制剂
维替泊芬（Visudyne），YAP抑制剂
$ 59.00
目录号 M60247
一种有效的选择性YAP抑制剂，可以破坏YAP-TEAD相互作用并增强YAP的胰蛋白酶切割。
VLX600，线粒体OXPHOS抑制剂VLX600，线粒体OXPHOS抑制剂
VLX600，线粒体OXPHOS抑制剂
$ 69.00
目录号 M60261
一种有效的和选择性的线粒体OXPHOS抑制剂。
VR23，蛋白酶体抑制剂VR23，蛋白酶体抑制剂
VR23，蛋白酶体抑制剂
$ 99.00
目录号 M60307
一种有效的和选择性的蛋白酶体抑制剂，其对胰蛋白酶样蛋白酶体，胰凝乳蛋白酶样蛋白酶体的IC50分别为1 nM，50-100 nM和3μM，
WAY-316606，分泌型卷曲蛋白相关蛋白-1（sFRP-1）抑制剂 WAY-316606，分泌型卷曲蛋白相关蛋白-1（sFRP-1）抑制剂
WAY-316606，分泌型卷曲蛋白相关蛋白-1（sFRP-1）抑制剂
$ 139.00
目录号 M60215
一种新型强效选择性分泌型卷曲相关蛋白-1（sFRP-1）抑制剂，可增加Wnt信号。
WDR5-0103，WDR5抑制剂WDR5-0103，WDR5抑制剂
WDR5-0103，WDR5抑制剂
$ 89.00
目录号 M60233
含有重复序列的WD重复蛋白5（WDR5）拮抗剂。
WDR5-C47，WDR5-MLL（SET1）拮抗剂 WDR5-C47，WDR5-MLL（SET1）拮抗剂
WDR5-C47，WDR5-MLL（SET1）拮抗剂
$ 129.00
目录号 M60118
WDR5-MLL相互作用的高度有效和选择性拮抗剂。
Wnt-C59，Wnt拮抗剂 Wnt-C59，Wnt拮抗剂
Wnt-C59，Wnt拮抗剂
$ 89.00
目录号 M60005
一种有效的，选择性和口服活性的Wnt信号通路拮抗剂。
WP1130（Degrasyn），去泛素化酶（DUB）抑制剂 WP1130（Degrasyn），去泛素化酶（DUB）抑制剂
WP1130（Degrasyn），去泛素化酶（DUB）抑制剂
$ 69.00
目录号 M60206
去泛素化酶（DUB）的细胞渗透性，有效和选择性抑制剂。
WS3，β细胞增殖诱导剂 WS3，β细胞增殖诱导剂
WS3，β细胞增殖诱导剂
$ 139.00
目录号 M60095 xcessbio小分子
一种高度有效和选择性的小分子，可促进胰腺β细胞和RPE细胞的扩增。
WS6，β细胞增殖诱导剂 WS6，β细胞增殖诱导剂
WS6，β细胞增殖诱导剂
$ 139.00
目录号 M60097
在啮齿动物和人类初级胰岛中促进胰腺β细胞增殖的高度有效和选择性的小分子，并显示极好的体内效力。
WWL113，Ces3和Ces1f抑制剂 WWL113，Ces3和Ces1f抑制剂
WWL113，Ces3和Ces1f抑制剂
$ 139.00
目录号 M60162
Ces3和Ces1f的新型有效和选择性抑制剂
XAV939 --- Wnt拮抗剂 XAV939 --- Wnt拮抗剂
XAV939 --- Wnt拮抗剂
$ 89.00
目录号 M60010
一种有效和选择性的Wnt途径拮抗剂; 通过抑制坦科聚合酶1和坦科聚合酶2来稳定axin。
XL888 --- HSP90抑制剂XL888 --- HSP90抑制剂
XL888 --- HSP90抑制剂
$ 149.00
目录号 M60164
一种高度有效的ATP竞争性和口服生物可利用的Hsp90抑制剂。
Y-27632 ---岩石抑制剂 Y-27632 ---岩石抑制剂
Y-27632 ---岩石抑制剂
$ 69.00
目录号 M60011
*广泛使用的岩石激酶抑制剂。
Y-320 --- IL-17**调节剂Y-320 --- IL-17**调节剂
Y-320 --- IL-17**调节剂
$ 89.00
目录号 M60200
一种口服有效的**调节剂，可抑制CD4T细胞对IL-15诱导的IL-17产生。
ZCL278 --- Cdc42 GTPase抑制剂ZCL278 --- Cdc42 GTPase抑制剂
ZCL278 --- Cdc42 GTPase抑制剂
$ 119.00
目录号 M60133
一种有效的选择性Cdc42 GTP酶抑制剂。
ZLN005 --- PGC-1α转录激活剂ZLN005 --- PGC-1α转录激活剂
ZLN005 --- PGC-1α转录激活剂
$ 69.00
目录号 M60142
一种有效和选择性的小分子PGC-1α转录激活剂。
